SCHEMBL8048477

SCHEMBL8048477

N=C(NCl)c1cccc(C(F)(F)F)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.55
NPSR1 Q6W5P4 1/20 0.47
P2RX1 P51575 1/20 0.47
LMNA P02545 1/20 0.47
SRD5A2 P31213 1/20 0.46
HTT P42858 1/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
ALDH1A1 P00352 1/20 0.45
POLB P06746 1/20 0.45
KCNK3 O14649 1/20 0.45
MAPT P10636 1/20 0.45
CNR1 P21554 1/20 0.44
TLR7 Q9NYK1 1/20 0.44
KCNQ3 O43525 1/20 0.44
KCNQ2 O43526 1/20 0.44
KCNE1 P15382 1/20 0.44
KCNQ1 P51787 1/20 0.44
KCNQ5 Q9NR82 1/20 0.44
PTGS1 P23219 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL642823 0.84 CES2 (0.56) CES2NPSR1P2RX1LMNASRD5A2
SCHEMBL4396979 0.82 CES2 (0.55) CES2NPSR1P2RX1LMNASRD5A2
Hydrochloric Acid SCHEMBL4400848 0.81 CES2 (0.53) CES2NPSR1P2RX1LMNASRD5A2
SCHEMBL3555007 0.79 CES2 (0.60) CES2NPSR1P2RX1LMNASRD5A2
SCHEMBL11553879 0.79 CES2 (0.51) CES2NPSR1P2RX1LMNASRD5A2
SCHEMBL10436303 0.79 CES2 (0.65) CES2NPSR1P2RX1LMNAHTT
SCHEMBL10285693 0.77 CES2 (0.48) CES2SRD5A2TLR7PTGS1
SCHEMBL15630195 0.77 CES2 (0.62) CES2NPSR1P2RX1LMNASRD5A2
SCHEMBL524006 0.76 CES2 (0.60) CES2SRD5A2PTGS1
SCHEMBL1826394 0.75 NPSR1 (0.55) CES2NPSR1P2RX1LMNASRD5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009068652-A1 2, 6-DISUBSTITUTED PYRIDINES AND 2, 4-DISUBSTITUTED PYRIMIDINES AS SOLUBLE GUANYLATE CYCLASE ACTIVATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed