SCHEMBL10285693

SCHEMBL10285693

N=C(NCl)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.48
CES1 P23141 2/20 0.48
SRD5A2 P31213 1/20 0.42
PTPN1 P18031 2/20 0.42
NR4A1 P22736 1/20 0.42
NR4A2 P43354 1/20 0.42
NR4A3 Q92570 1/20 0.42
GSK3B P49841 2/20 0.41
TRPV1 Q8NER1 2/20 0.40
PTGS1 P23219 2/20 0.40
MMP1 P03956 1/20 0.40
EPHX2 P34913 1/20 0.39
TLR7 Q9NYK1 1/20 0.39
IDO1 P14902 1/20 0.39
ORAI1 Q96D31 1/20 0.39
ORAI2 Q96SN7 1/20 0.39
ORAI3 Q9BRQ5 1/20 0.39
TRPV6 Q9H1D0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2314418 0.81 CES2 (0.50) CES2CES1SRD5A2PTPN1GSK3B
SCHEMBL4399783 0.79 CES2 (0.48) CES2CES1SRD5A2PTPN1GSK3B
SCHEMBL30388464 0.79 CES2 (0.48) CES2CES1SRD5A2PTPN1NR4A1
Hydrochloric Acid SCHEMBL4394743 0.78 CES2 (0.47) CES2CES1SRD5A2PTPN1GSK3B
SCHEMBL8048477 0.77 CES2 (0.55) CES2SRD5A2PTGS1TLR7
SCHEMBL8578258 0.77 CES2 (0.61) CES2CES1SRD5A2PTPN1NR4A1
SCHEMBL5206631 0.76 CES2 (0.54) CES2CES1SRD5A2PTPN1NR4A1
SCHEMBL1005632 0.75 CES2 (0.58) CES2CES1SRD5A2PTPN1NR4A1
SCHEMBL28415675 0.73 RAB9A (0.57) TRPV1PTGS1EPHX2
SCHEMBL20946216 0.72 MAPK14 (0.47) CES2CES1TRPV1MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120053053-A1 PYRIMIDINE DERIVATIVES AND THEIR USE AS HERBICIDES SYNGENTA CROP PROTECTION, LLC (US) 2012-03-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120053053-A1 PYRIMIDINE DERIVATIVES AND THEIR USE AS HERBICIDES DPYD, DHODH, TYMP CES2 1575/4885CES1 1371/4885SRD5A2 983/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.