SCHEMBL8048882

SCHEMBL8048882

COc1ccc2c(c1)CC[C@@H]1[C@@H]3CC[C@@H](CC(=O)O)[C@@]3(C)CC[C@]21O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 2/20 0.42
POLA1 P09884 2/20 0.41
ESR1 P03372 2/20 0.39
LMNA P02545 2/20 0.39
HSD17B10 Q99714 1/20 0.39
KDM1A O60341 1/20 0.38
MAPT P10636 1/20 0.37
HSD17B1 P14061 1/20 0.37
RECQL P46063 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
FFAR4 Q5NUL3 1/20 0.37
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
ESR2 Q92731 1/20 0.36
CYP2C19 P33261 2/20 0.36
CYP2C9 P11712 1/20 0.36
TSHR P16473 1/20 0.36
CYP3A4 P08684 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8048886 1.00 PPARD (0.42) PPARDPOLA1ESR1LMNAHSD17B10
SCHEMBL8049873 1.00 PPARD (0.42) PPARDPOLA1ESR1LMNAHSD17B10
SCHEMBL8049867 1.00 PPARD (0.42) PPARDPOLA1ESR1LMNAHSD17B10
SCHEMBL8052780 0.86 PPARD (0.41) PPARDPOLA1ESR1LMNAKDM1A
SCHEMBL7515670 0.84 PPARD (0.38) PPARDPOLA1ESR1LMNAHSD17B10
SCHEMBL8048425 0.82 LMNA (0.56) ESR1LMNAHSD17B10KDM1AMAPT
SCHEMBL8048890 0.82 LMNA (0.56) ESR1LMNAHSD17B10KDM1AMAPT
SCHEMBL11222251 0.76 STS (0.60) POLA1ESR1LMNAHSD17B10MAPT
SCHEMBL11671496 0.76 STS (0.60) POLA1ESR1LMNAHSD17B10MAPT
SCHEMBL8048295 0.76 STS (0.60) POLA1ESR1LMNAHSD17B10MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0882735-B1 9 Alpha-hydroxy-8 alpha-estra-1,3,5(10)-trienes and a process for their preparation JENAPHARM GMBH (DE) 2000-04-19 EP disclosed
EP-0882735-A1 9 Alpha-hydroxy-8 alpha-estra-1,3,5(10)-trienes and a process for their preparation Jenapharm GmbH & Co. KG (DE) 1998-12-09 EP disclosed