SCHEMBL8050331

SCHEMBL8050331

FC(F)(F)c1ccc(-c2nnc(S)s2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 4/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
NPC1 O15118 3/20 0.42
RAB9A P51151 2/20 0.42
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
QPCT Q16769 3/20 0.40
QPCTL Q9NXS2 1/20 0.40
MAPT P10636 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
P2RY1 P47900 1/20 0.38
S1PR1 P21453 1/20 0.38
MAOB P27338 1/20 0.37
MEN1 O00255 1/20 0.37
HSP90AA1 P07900 1/20 0.37
CRHBP P24387 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14557099 0.84 KDM4E (0.43) NPC1RAB9AKDM4EALDH1A1GAA
SCHEMBL8044533 0.81 IKBKB (0.36) HDAC1HDAC2ALDH1A1QPCTSMN1; SMN2
SCHEMBL20214353 0.78 KDM4E (0.69) KIF11NPC1RAB9AKDM4EALDH1A1
SCHEMBL20214059 0.78 KDM4E (0.46) KIF11HDAC1HDAC2NPC1RAB9A
SCHEMBL8048162 0.77 P2RY1 (0.41) KIF11NPC1RAB9AKDM4EALDH1A1
SCHEMBL969939 0.76 KDM4E (0.59) NPC1RAB9AKDM4EALDH1A1GAA
SCHEMBL20214047 0.75 HDAC1 (0.51) KIF11HDAC1HDAC2NPC1RAB9A
SCHEMBL8047389 0.75 CA1 (0.49) HDAC1HDAC2NPC1RAB9AKDM4E
SCHEMBL28353374 0.75 ALDH1A1 (0.48) NPC1RAB9AKDM4EALDH1A1GAA
SCHEMBL9360268 0.75 GAA (0.60) HDAC1HDAC2NPC1RAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104292224-B Containing replacing 1,3,4-thiophene () diazole thioether benzothiazole amide derivatives and its preparation method and application 贵州大学 2016-07-06 CN disclosed
CN-104292224-A Benzothiazole amide derivatives containing substituted 1,3,4-thiadiazole (oxadiazole) thioether as well as preparation method and application of derivatives UNIV GUIZHOU 2015-01-21 CN disclosed
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed