SCHEMBL8044533

SCHEMBL8044533

FC(F)(F)c1cc(-c2nnc(S)s2)cc(C(F)(F)F)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.36
F2RL3 Q96RI0 1/20 0.33
RXRA P19793 2/20 0.33
RXRB P28702 2/20 0.33
RXRG P48443 2/20 0.33
PIM1 P11309 2/20 0.32
CDK1 P06493 1/20 0.32
CDK2 P24941 1/20 0.32
MAPKAPK2 P49137 1/20 0.32
GSK3A P49840 1/20 0.32
GSK3B P49841 1/20 0.32
CDK5 Q00535 1/20 0.32
DYRK1A Q13627 1/20 0.32
PIM3 Q86V86 1/20 0.32
CES2 O00748 1/20 0.31
S1PR1 P21453 1/20 0.31
S1PR3 Q99500 1/20 0.31
CNR1 P21554 2/20 0.30
CNR2 P34972 2/20 0.30
QPCT Q16769 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8050331 0.81 KIF11 (0.44) S1PR1QPCTHDAC1HDAC2ALDH1A1
SCHEMBL14557095 0.80 SNCA (0.37) PTGS1PTGS2ALDH1A1SMN1; SMN2
SCHEMBL969945 0.71 PIK3CA (0.40) PTGS1PTGS2ALDH1A1SMN1; SMN2
SCHEMBL14557099 0.71 KDM4E (0.43) ALDH1A1SMN1; SMN2
SCHEMBL14338261 0.68 CES2 (0.48) IKBKBRXRARXRBRXRGCES2
SCHEMBL9482063 0.67 RXRA (0.54) IKBKBRXRARXRBRXRGCES2
SCHEMBL8050989 0.67 ALDH1A1 (0.60) PTGS2HDAC1HDAC2ALDH1A1SMN1; SMN2
SCHEMBL8048162 0.67 P2RY1 (0.41) F2RL3ALDH1A1SMN1; SMN2
SCHEMBL2753490 0.67 IKBKB (0.36) IKBKBF2RL3RXRARXRBRXRG
SCHEMBL8046027 0.67 CYP1A1 (0.46) PTGS1PTGS2ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed