SCHEMBL8053422

SCHEMBL8053422

CC(C)CN(c1ccncc1)c1csc2cc(Cl)ccc12

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.35
CYP2A6 P11509 2/20 0.33
AKT1 P31749 1/20 0.33
SLC6A2 P23975 1/20 0.31
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8053832 0.99 ROCK1 (0.34) ROCK1CYP2A6AKT1SLC6A2NOS3
SCHEMBL8050470 0.86 ROCK1 (0.37) ROCK1CYP2A6SLC6A2NOS3NOS1
Hydrochloric Acid SCHEMBL8051640 0.85 ROCK1 (0.36) ROCK1CYP2A6SLC6A2NOS3NOS1
SCHEMBL8056707 0.84 SLC6A2 (0.41) ROCK1CYP2A6SLC6A2NOS3NOS1
SCHEMBL8050534 0.83 ROCK1 (0.35) ROCK1CYP2A6SLC6A2NOS3NOS1
Hydrochloric Acid SCHEMBL8038855 0.83 SLC6A2 (0.40) ROCK1CYP2A6SLC6A2NOS3NOS1
SCHEMBL8050015 0.82 POLQ (0.35) SLC6A2
SCHEMBL8053815 0.82 ROCK1 (0.41) ROCK1CYP2A6AKT1SLC6A2
SCHEMBL8051666 0.82 ALDH1A1 (0.37) CYP2A6AKT1SLC6A2
SCHEMBL8039432 0.82 SLC6A2 (0.37) ROCK1CYP2A6SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6022880-A Substituted pyridylamino indoles HOECHST MARION ROUSSEL, INC. (US) 2000-02-08 US disclosed
US-5328920-A Alleviating memory dysfunctions HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1994-07-12 US disclosed