SCHEMBL8055265

SCHEMBL8055265

Cc1ccc2ccocc1-2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.39
LPL P06858 1/20 0.36
LIPG Q9Y5X9 1/20 0.36
ALDH1A1 P00352 2/20 0.35
IMPDH2 P12268 2/20 0.34
MAPK14 Q16539 2/20 0.34
HSPB1 P04792 1/20 0.34
ESR2 Q92731 1/20 0.33
PTGER2 P43116 1/20 0.33
ENPP3 O14638 1/20 0.33
ENPP1 P22413 1/20 0.33
ERN1 O75460 1/20 0.32
CHEK1 O14757 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA9 Q16790 1/20 0.31
FYN P06241 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7696358 0.81 IMPDH2 (0.38) LPLLIPGALDH1A1IMPDH2MAPK14
SCHEMBL14003430 0.74 S1PR4 (0.39) ALDH1A1IMPDH2CYP1A2CYP3A4CYP2D6
SCHEMBL2010826 0.71 ESR1 (0.39) ESR1LPLLIPGALDH1A1IMPDH2
SCHEMBL10304989 0.71 ABL1 (0.41) ALDH1A1IMPDH2LMNACYP1A2CYP3A4
SCHEMBL20777196 0.71 CSNK2A1 (0.41) IMPDH2ADORA3CYP3A4CSNK2A1
SCHEMBL5795534 0.71 ALDH1A1 (0.43) ALDH1A1IMPDH2FYNLMNACYP3A4
SCHEMBL6980495 0.70 ALDH1A1 (0.44) ESR1ALDH1A1IMPDH2ESR2FYN
SCHEMBL10035040 0.69 PPARG (0.48) ALDH1A1ERN1FYNLMNACYP1A2
SCHEMBL20036777 0.69 TOP2A (0.38) ESR1LPLLIPGALDH1A1IMPDH2
SCHEMBL11483469 0.69 PTGER2 (0.38) ESR1LPLLIPGPTGER2ERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105492437-A Substituted benzofuranyl and benzoxazolyl compounds and uses thereof KARYOPHARM THERAPEUTICS INC 2016-04-13 CN disclosed
US-6040449-A USEFUL FOR FORMING FLUORINE CONTAINING 1,4-DISUBSTITUTED PIPERIDINE DERIVATIVES, USEFUL AS ANTAGONIST FOR MUSCARINIC M3 RECEPTORS AND LESS SIDE EFFECT BANYU PHARMACEUTICAL CO LTD (JP) 2000-03-21 US disclosed
US-5948792-A POTENT AND SELECTIVE ANTAGONISTS FOR MUSCARINIC M.SUB.3 RECEPTORS WITH LITTLE SIDE EFFECTS. BANYU PHARMACEUTICAL CO., LTD. (JP) 1999-09-07 US disclosed
EP-0930298-A1 FLUORINATED 1,4-DISUBSTITUTED PIPERIDINE DERIVATIVES BANYU PHARMACEUTICAL CO., LTD. (JP) 1999-07-21 EP disclosed