SCHEMBL8055301

SCHEMBL8055301

CCc1nc(Br)cnc1CCN

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCR4 P51679 1/20 0.35
HRH1 P35367 2/20 0.35
HRH4 Q9H3N8 2/20 0.35
HRH2 P25021 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
TDP1 Q9NUW8 1/20 0.34
TAAR1 Q96RJ0 1/20 0.32
EDNRA P25101 1/20 0.32
CHEK1 O14757 1/20 0.31
CCNA2 P20248 1/20 0.31
CDK2 P24941 1/20 0.31
CCNA1 P78396 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27501035 0.77 CCR4 (0.33) CCR4EDNRA
SCHEMBL8055545 0.76 CCR4 (0.38) CCR4TDP1EDNRA
SCHEMBL30427027 0.76 CCR4 (0.38) CCR4TDP1EDNRA
SCHEMBL11229329 0.74 CCR4 (0.39) CCR4EDNRA
SCHEMBL11223843 0.73 CCR4 (0.35) CCR4EDNRA
SCHEMBL11223672 0.71 CCR4 (0.38) CCR4EDNRA
SCHEMBL10271758 0.68 CCR4 (0.40) CCR4EDNRA
SCHEMBL23250599 0.67 CCR4 (0.38) CCR4EDNRA
SCHEMBL29862850 0.67 CCR4 (0.38) CCR4EDNRA
SCHEMBL7418341 0.66 HTT (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6083951-A FOR THE TREATMENT OF DISEASES OR MEDICAL CONDITIONS SUCH AS HYPERTENSION, PULMONARY HYPERTENSION, CARDIAC OR CEREBRAL CIRCULATORY DISEASE AND RENAL DISEASE ZENECA LIMITED (GB) 2000-07-04 US disclosed