SCHEMBL8055688

SCHEMBL8055688

COc1ccc([CH]C2CC2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.50
CYP2A6 P11509 1/20 0.50
KDM4E B2RXH2 4/20 0.48
CYP3A4 P08684 2/20 0.48
LMNA P02545 2/20 0.48
TP53 P04637 1/20 0.48
TSHR P16473 1/20 0.48
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA7 P43166 1/20 0.48
CA9 Q16790 1/20 0.48
CA14 Q9ULX7 1/20 0.48
TRPA1 O75762 1/20 0.47
RELA Q04206 1/20 0.47
CHRNA7 P36544 1/20 0.46
CYP1A2 P05177 4/20 0.45
CYP1A1 P04798 3/20 0.45
CYP1B1 Q16678 3/20 0.45
ESR1 P03372 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4494269 0.75 ALDH1A1 (0.47) ALDH1A1CYP2A6KDM4ECYP3A4LMNA
SCHEMBL3019888 0.75 CYP2A6 (0.44) ALDH1A1CYP2A6KDM4ETSHRCA1
SCHEMBL4518823 0.74 PIM1 (0.45) ALDH1A1KDM4EMAPTCYP2D6MAOB
SCHEMBL14329775 0.74 RELA (0.67) ALDH1A1KDM4ECYP3A4LMNATP53
SCHEMBL6301892 0.72 HPGD (0.44) ALDH1A1CYP2A6KDM4ECYP3A4LMNA
SCHEMBL9292663 0.72 MAOB (0.55) ALDH1A1KDM4ECYP3A4LMNATP53
SCHEMBL9292660 0.72 MAOB (0.55) ALDH1A1KDM4ECYP3A4LMNATP53
SCHEMBL9292664 0.72 MAOB (0.55) ALDH1A1KDM4ECYP3A4LMNATP53
SCHEMBL23020629 0.72 MAOB (0.58) ALDH1A1CYP2A6KDM4ECYP3A4LMNA
SCHEMBL2449268 0.72 KDM4E (0.70) ALDH1A1CYP2A6KDM4ECYP3A4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6037340-A HAVE BIOLOGICAL ACTIVITY INCLUDING ANTI-CANCER ACTIVITY CADUS PHARMACEUTICAL CORPORATION (US) 2000-03-14 US disclosed
WO-1998054116-A1 SYNTHESIS AND USE OF THIOPHENE- AND PYRROLE-BASED HETEROAROMATIC COMPOUNDS CADUS PHARMACEUTICAL CORPORATION (US) 1998-12-03 WO disclosed
WO-1995023784-A1 CARBAMOYL CARBOXYLIC ACID AMIDES, PROCESS FOR PRODUCING THEM AND THEIR USE AS FUNGICIDES BASF AKTIENGESELLSCHAFT (DE) 1995-09-08 WO disclosed