SCHEMBL8056997

SCHEMBL8056997

COC(=O)c1ccc2c(c1)S(=O)(=O)CC(C)(C)C2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
XDH P47989 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
KDM4E B2RXH2 7/20 0.41
MAPT P10636 3/20 0.41
TRPA1 O75762 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
HSD17B10 Q99714 3/20 0.39
PDK2 Q15119 2/20 0.39
POLB P06746 1/20 0.39
ALDH1A1 P00352 8/20 0.39
GAA P10253 2/20 0.39
EGFR P00533 1/20 0.39
ERBB2 P04626 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8045106 0.81 ALDH1A1 (0.35) CA12CA1CA2CA7CA9
SCHEMBL8062898 0.79 CYP3A4 (0.44) CA12CA1CA2CA7XDH
SCHEMBL8060684 0.79 CA1 (0.44) CA12CA1CA2CA7XDH
SCHEMBL8045175 0.79 HTR7 (0.44)
SCHEMBL8056289 0.78 ALDH1A1 (0.46) CA12CA1CA2CA7XDH
SCHEMBL8058029 0.77 PDK2 (0.42) CA12CA1CA2CA7XDH
SCHEMBL8057407 0.76 PDK2 (0.41) CA12CA1CA2CA7XDH
SCHEMBL8060825 0.76 PDK2 (0.41) CA12CA1CA2CA7XDH
SCHEMBL8060786 0.76 CA1 (0.46) CA12CA1CA2CA7XDH
SCHEMBL8057016 0.76 ALDH1A1 (0.35) KDM4EMAPTHSD17B10POLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed