SCHEMBL8062898

SCHEMBL8062898

COC(=O)c1ccc2c(c1)S(=O)(=O)CC2(C)C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.44
PDK2 Q15119 2/20 0.44
CA12 O43570 2/20 0.44
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
CA7 P43166 2/20 0.44
CA9 Q16790 2/20 0.44
CA14 Q9ULX7 2/20 0.44
XDH P47989 1/20 0.44
ALDH1A1 P00352 5/20 0.43
PTPN11 Q06124 1/20 0.42
RARA P10276 1/20 0.41
RARB P10826 1/20 0.41
RARG P13631 1/20 0.41
CYP26A1 O43174 2/20 0.41
KDM4E B2RXH2 4/20 0.41
MAPT P10636 2/20 0.41
HPGD P15428 2/20 0.41
HSD17B10 Q99714 2/20 0.41
GLA P06280 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8056289 0.87 ALDH1A1 (0.46) CYP3A4PDK2CA12CA1CA2
SCHEMBL8058029 0.85 PDK2 (0.42) CYP3A4PDK2CA12CA1CA2
SCHEMBL8056479 0.85 CYP3A4 (0.48) CYP3A4PDK2CA12CA1CA2
SCHEMBL3275738 0.84 RARB (0.46) CYP3A4ALDH1A1RARARARBRARG
SCHEMBL8057407 0.84 PDK2 (0.41) CYP3A4PDK2CA12CA1CA2
SCHEMBL8060825 0.84 PDK2 (0.41) CYP3A4PDK2CA12CA1CA2
SCHEMBL8058171 0.82 PDK2 (0.40) CYP3A4PDK2CA12CA1CA2
SCHEMBL8045253 0.80 ALDH1A1 (0.43) PDK2CA12CA1CA2CA7
SCHEMBL8056997 0.79 CA12 (0.41) PDK2CA12CA1CA2CA7
SCHEMBL8058138 0.79 KDM4E (0.36) ALDH1A1RARARARBRARGKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed