SCHEMBL8057262

SCHEMBL8057262

O=C(NC1CCN(CCN2CCNCC2)CC1)c1n[nH]c2ccccc12

nearest known ligand 0.65

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.65
RAB9A P51151 1/20 0.65
SMYD3 Q9H7B4 1/20 0.60
USP30 Q70CQ3 1/20 0.60
DYRK1A Q13627 7/20 0.56
WNT1 P04628 5/20 0.56
CHRNA7 P36544 5/20 0.55
HTR3A P46098 2/20 0.55
HTR1A P08908 2/20 0.53
DRD2 P14416 2/20 0.53
HTR2A P28223 2/20 0.53
FLT3 P36888 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6951767 0.86 NPC1 (0.64) NPC1RAB9ASMYD3USP30DYRK1A
SCHEMBL4384530 0.86 NPC1 (0.82) NPC1RAB9ASMYD3USP30DYRK1A
SCHEMBL6954648 0.84 HTR1A (0.65) NPC1RAB9AHTR1ADRD2HTR2A
SCHEMBL6950689 0.84 NPC1 (0.74) NPC1RAB9ASMYD3USP30DYRK1A
SCHEMBL29732688 0.84 NPC1 (0.74) NPC1RAB9ASMYD3USP30DYRK1A
SCHEMBL3164026 0.83 WNT1 (0.69) NPC1RAB9ASMYD3USP30DYRK1A
SCHEMBL8162625 0.83 NPC1 (0.65) NPC1RAB9ASMYD3USP30DYRK1A
SCHEMBL6951433 0.80 NPC1 (0.68) NPC1RAB9ASMYD3USP30DYRK1A
SCHEMBL7376957 0.80 RAB9A (0.54) NPC1RAB9ASMYD3USP30DYRK1A
SCHEMBL26400414 0.79 NPC1 (0.97) NPC1RAB9ASMYD3USP30DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6117882-A 5-HT4 agonists and antagonists ELI LILLY AND COMPANY (US) 2000-09-12 US disclosed
US-6069152-A NERVOUS SYSTEM DISORDERS; CARDIOVASCULAR DISORDERS; GASTROINTESTINAL DISORDERS ELI LILLY AND COMPANY (US) 2000-05-30 US disclosed
EP-0908459-A1 5-HT4 Agonists and antagonists ELI LILLY AND COMPANY (US) 1999-04-14 EP disclosed