SCHEMBL8057965

SCHEMBL8057965

CCCCOc1cc(C2SCCCS2)ccc1OC

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.53
PDE4A P27815 9/20 0.53
PDE4D Q08499 5/20 0.53
PDE4B Q07343 4/20 0.53
PDE4C Q08493 4/20 0.53
MAPK1 P28482 2/20 0.43
TNF P01375 1/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
PDE3B Q13370 1/20 0.43
PDE3A Q14432 1/20 0.43
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
NFKB1 P19838 1/20 0.43
KMT2A Q03164 1/20 0.43
SMPD1 P17405 4/20 0.40
MPO P05164 1/20 0.39
FPR2 P25090 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8064807 0.95 TSHR (0.53) TSHRPDE4APDE4DPDE4BPDE4C
SCHEMBL8059997 0.93 TSHR (0.47) TSHRPDE4APDE4DPDE4BPDE4C
SCHEMBL8058003 0.90 TSHR (0.51) TSHRPDE4APDE4DPDE4BPDE4C
SCHEMBL3757194 0.88 TSHR (0.45) TSHRPDE4APDE4DPDE4BPDE4C
SCHEMBL9778850 0.87 TSHR (0.57) TSHRPDE4APDE4DPDE4BPDE4C
SCHEMBL30669513 0.84 TSHR (0.67) TSHRPDE4APDE4DPDE4BPDE4C
SCHEMBL8057984 0.84 TSHR (0.67) TSHRPDE4APDE4DPDE4BPDE4C
SCHEMBL8059968 0.84 TSHR (0.47) TSHRPDE4APDE4DPDE4BPDE4C
SCHEMBL9778782 0.82 TSHR (0.57) TSHRPDE4AMAPK1MAPTKDM4E
SCHEMBL9778817 0.80 TSHR (0.50) TSHRPDE4AMAPTKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1004623-A1 Aryl thioacetals useful as stabilizers in polymeric materials GREAT LAKES CHEMICAL CORPORATION (US) 2000-05-31 EP disclosed
US-4127588-A Sulphur containing derivatives HOFFMANN-LA ROCHE INC. (US) 1978-11-28 US disclosed
US-4073797-A CORONARY DILATOR HOFFMANN-LA ROCHE INC. (US) 1978-02-14 US disclosed
US-4003914-A DITHIANE AND DISULFONE CORONARY DILATING AGENTS HOFFMANN-LA ROCHE INC. (US) 1977-01-18 US disclosed