SCHEMBL8058007

SCHEMBL8058007

CON=C1CS(=O)(=O)c2cc(C(=O)OC)c(F)cc21

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.35
SOS1 Q07889 1/20 0.33
ALDH1A1 P00352 2/20 0.31
HPGD P15428 2/20 0.31
HSD17B10 Q99714 2/20 0.31
PDK2 Q15119 2/20 0.31
TSHR P16473 1/20 0.31
ALPL P05186 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
PKLR P30613 1/20 0.30
PKM P14618 1/20 0.30
GAA P10253 2/20 0.30
KDM4E B2RXH2 1/20 0.30
GLA P06280 1/20 0.30
MAPT P10636 1/20 0.30
CASP1 P29466 1/20 0.30
CASP7 P55210 1/20 0.30
ATM Q13315 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8058006 1.00 CTSL (0.35) CTSLSOS1ALDH1A1HPGDHSD17B10
SCHEMBL8056507 0.88 CTSL (0.36) CTSLALDH1A1HPGDHSD17B10PDK2
SCHEMBL8056511 0.88 CTSL (0.36) CTSLALDH1A1HPGDHSD17B10PDK2
SCHEMBL8056913 0.86 ALDH1A1 (0.33) ALDH1A1HPGDHSD17B10TSHRSLC6A3
SCHEMBL8056918 0.86 ALDH1A1 (0.33) ALDH1A1HPGDHSD17B10TSHRSLC6A3
SCHEMBL8056935 0.84
SCHEMBL8056931 0.84
SCHEMBL8058223 0.84 CFTR (0.37) SOS1PDK2MAPT
SCHEMBL8058221 0.84 CFTR (0.37) SOS1PDK2MAPT
SCHEMBL8060841 0.84 CTSL (0.32) CTSLALDH1A1HPGDHSD17B10TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed