SCHEMBL8058060

SCHEMBL8058060

COc1cc(N)c(Cl)cc1C(=O)NC1(CN2CCC(C)CC2)CCCCC1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 7/20 0.58
HTR3A P46098 2/20 0.56
HTR3E A5X5Y0 1/20 0.56
HTR3B O95264 1/20 0.56
HTR3D Q70Z44 1/20 0.56
HTR3C Q8WXA8 1/20 0.56
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
ADRA2A P08913 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
DRD2 P14416 1/20 0.52
ADRA2B P18089 1/20 0.52
ADRA2C P18825 1/20 0.52
DRD4 P21917 1/20 0.52
ACHE P22303 1/20 0.52
SLC6A2 P23975 1/20 0.52
HTR2A P28223 1/20 0.52
HTR2C P28335 1/20 0.52
ADRA1A P35348 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8040144 0.92 HTR4 (0.57) HTR4HTR3AHTR3EHTR3BHTR3D
SCHEMBL8055027 0.91 HTR4 (0.64) HTR4HTR3AHTR3EHTR3BHTR3D
SCHEMBL8054707 0.91 HTR4 (0.53) HTR4HTR3AHTR3EHTR3BHTR3D
SCHEMBL8040211 0.90 CNR2 (0.47) HTR4HTR3AHTR3EHTR3BHTR3D
SCHEMBL8040220 0.90 HTR4 (0.58) HTR4HTR3AHTR3EHTR3BHTR3D
SCHEMBL8054528 0.86 DRD4 (0.53) DRD2DRD4DRD3
SCHEMBL8050559 0.82 CNR2 (0.50) HTR4HTR3AHTR3EHTR3BHTR3D
SCHEMBL8051399 0.81 CNR2 (0.48) HTR4HTR3AHTR3EHTR3BHTR3D
SCHEMBL8051372 0.78 DRD4 (0.54) DRD2DRD4DRD3
SCHEMBL8039975 0.77 DRD4 (0.50) HTR4HTR3AHTR3EHTR3BHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0998469-A1 BENZAMIDE CYCLOALKYL STIMULATING HIGH AND LOW GASTROINTESTINAL MOTRICITY Laboratoires Jacques Logeais (FR) 2000-05-10 EP disclosed
WO-1999005133-A1 BENZAMIDE CYCLOALKYL STIMULATING HIGH AND LOW GASTROINTESTINAL MOTRICITY LABORATOIRES JACQUES LOGEAIS (FR) 1999-02-04 WO disclosed