SCHEMBL8040211

SCHEMBL8040211

CC1CCN(CC2(NC(=O)c3cc(Cl)c(N)cc3OCC3CC3)CCCCC2)CC1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.47
HTR4 Q13639 9/20 0.47
ACHE P22303 2/20 0.45
HTR3E A5X5Y0 1/20 0.45
HTR3B O95264 1/20 0.45
HTR3A P46098 1/20 0.45
HTR3D Q70Z44 1/20 0.45
HTR3C Q8WXA8 1/20 0.45
DRD2 P14416 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8050559 0.93 CNR2 (0.50) CNR2HTR4ACHEHTR3EHTR3B
SCHEMBL8054707 0.92 HTR4 (0.53) HTR4ACHEHTR3EHTR3BHTR3A
SCHEMBL8051399 0.92 CNR2 (0.48) CNR2HTR4ACHEHTR3EHTR3B
SCHEMBL8058060 0.90 HTR4 (0.58) HTR4ACHEHTR3EHTR3BHTR3A
SCHEMBL8040144 0.82 HTR4 (0.57) HTR4ACHEHTR3EHTR3BHTR3A
SCHEMBL8055027 0.81 HTR4 (0.64) HTR4HTR3EHTR3BHTR3AHTR3D
SCHEMBL8040220 0.80 HTR4 (0.58) HTR4ACHEHTR3EHTR3BHTR3A
Lirexapride SCHEMBL384567 0.78 HTR4 (0.50) HTR4ACHEDRD2
SCHEMBL8052736 0.77 HTR4 (0.52) HTR4
SCHEMBL8054528 0.77 DRD4 (0.53) DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0998469-A1 BENZAMIDE CYCLOALKYL STIMULATING HIGH AND LOW GASTROINTESTINAL MOTRICITY Laboratoires Jacques Logeais (FR) 2000-05-10 EP disclosed
WO-1999005133-A1 BENZAMIDE CYCLOALKYL STIMULATING HIGH AND LOW GASTROINTESTINAL MOTRICITY LABORATOIRES JACQUES LOGEAIS (FR) 1999-02-04 WO disclosed