SCHEMBL8058138

SCHEMBL8058138

COC(=O)c1cc2c(cc1C)C(C)(C)CS2(=O)=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.36
ALDH1A1 P00352 6/20 0.36
HSD17B10 Q99714 3/20 0.36
HPGD P15428 2/20 0.36
MAPT P10636 2/20 0.36
GAA P10253 2/20 0.36
GLA P06280 1/20 0.36
CASP1 P29466 1/20 0.36
CASP7 P55210 1/20 0.36
ATM Q13315 1/20 0.36
RARA P10276 2/20 0.35
RARB P10826 2/20 0.35
RARG P13631 2/20 0.35
RXRA P19793 4/20 0.34
RXRB P28702 4/20 0.34
RXRG P48443 4/20 0.34
PDGFRB P09619 1/20 0.34
FGFR1 P11362 1/20 0.34
PDGFRA P16234 1/20 0.34
FLT1 P17948 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8062941 0.87 KDM4E (0.35) KDM4EALDH1A1HSD17B10HPGDMAPT
SCHEMBL8045223 0.86 RXRA (0.38) RARARARBRARGRXRARXRB
SCHEMBL8045039 0.84 RARB (0.35) KDM4EALDH1A1HSD17B10HPGDMAPT
SCHEMBL8062746 0.83 RXRA (0.36) KDM4EALDH1A1HSD17B10HPGDMAPT
SCHEMBL8045123 0.82 KDM4E (0.33) KDM4EALDH1A1HSD17B10HPGDMAPT
SCHEMBL8058195 0.81 CFTR (0.39) MAPT
SCHEMBL8062769 0.81 PDGFRA (0.34) KDM4EALDH1A1HSD17B10HPGDMAPT
SCHEMBL8060665 0.81 ALDH1A1 (0.36) KDM4EALDH1A1HSD17B10HPGDMAPT
SCHEMBL8062898 0.79 CYP3A4 (0.44) KDM4EALDH1A1HSD17B10HPGDMAPT
SCHEMBL8045106 0.78 ALDH1A1 (0.35) KDM4EALDH1A1HSD17B10HPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed