SCHEMBL8058145

SCHEMBL8058145

CCc1cc2c(cc1C(=O)OC)S(=O)(=O)CC2=NO

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.32
ALDH1A1 P00352 6/20 0.32
MAPT P10636 4/20 0.32
KDM4E B2RXH2 4/20 0.32
HTT P42858 2/20 0.32
HSD17B10 Q99714 2/20 0.32
TSHR P16473 2/20 0.32
MEN1 O00255 1/20 0.32
MAPK10 P53779 1/20 0.32
KMT2A Q03164 1/20 0.32
PTK2B Q14289 1/20 0.32
NCOA1 Q15788 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
NCOA3 Q9Y6Q9 1/20 0.32
POLB P06746 1/20 0.31
HPGD P15428 2/20 0.31
LMNA P02545 2/20 0.31
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8058144 1.00 CTSL (0.32) CTSLALDH1A1MAPTKDM4EHTT
SCHEMBL8060842 0.89 CTSL (0.32) CTSLALDH1A1MAPTKDM4EHTT
SCHEMBL8060841 0.89 CTSL (0.32) CTSLALDH1A1MAPTKDM4EHTT
SCHEMBL8056990 0.84 KDM4E (0.34) ALDH1A1MAPTKDM4EHTTHSD17B10
SCHEMBL8056988 0.84 KDM4E (0.34) ALDH1A1MAPTKDM4EHTTHSD17B10
SCHEMBL8056511 0.83 CTSL (0.36) CTSLALDH1A1MAPTKDM4EHTT
SCHEMBL8056507 0.83 CTSL (0.36) CTSLALDH1A1MAPTKDM4EHTT
SCHEMBL8045172 0.83 VEGFA (0.35) ALDH1A1MAPTKDM4EHTTHSD17B10
SCHEMBL8062968 0.82 ALDH1A1 (0.33) ALDH1A1MAPTKDM4EHTTHSD17B10
SCHEMBL8056235 0.80 CFTR (0.38) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed