SCHEMBL8058760

SCHEMBL8058760

O=C(Nc1ccc(Cl)cc1)N[C@@H](c1ccccc1)[C@@H](NC(=O)NC1CCCCC1)c1ccccc1

nearest known ligand 0.67

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 11/20 0.67
RAB9A P51151 9/20 0.67
NPC1 O15118 7/20 0.67
SMN1; SMN2 Q16637 4/20 0.67
ALDH1A1 P00352 1/20 0.67
CYP2C9 P11712 1/20 0.67
CYP2C19 P33261 1/20 0.67
EPHX2 P34913 5/20 0.59
LMNA P02545 2/20 0.56
TP53 P04637 1/20 0.56
NFKB1 P19838 1/20 0.56
NFKB2 Q00653 1/20 0.56
RELA Q04206 1/20 0.56
CNR1 P21554 2/20 0.53
MEN1 O00255 2/20 0.52
TSHR P16473 2/20 0.52
KMT2A Q03164 2/20 0.52
GAA P10253 1/20 0.50
HTT P42858 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8058763 1.00 EPHX1 (0.67) EPHX1RAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL8069606 0.87 RAB9A (0.72) EPHX1RAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL8069608 0.87 RAB9A (0.72) EPHX1RAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL8067568 0.86 EPHX1 (0.73) EPHX1RAB9ANPC1SMN1; SMN2CYP2C19
SCHEMBL8058426 0.85 EPHX1 (0.70) EPHX1RAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL8058429 0.85 EPHX1 (0.70) EPHX1RAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL8069610 0.84 EPHX1 (0.70) EPHX1RAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL8069612 0.84 EPHX1 (0.70) EPHX1RAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL8067991 0.83 RAB9A (0.72) EPHX1RAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL8067993 0.83 RAB9A (0.72) EPHX1RAB9ANPC1SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6103761-A Agents acting at cholecystokinin receptors WARNER-LAMBERT COMPANY (US) 2000-08-15 US disclosed
US-5389682-A Appetite suppressants, anxiolytic agents, gastric acid inhibition WARNER-LAMBERT COMPANY (US) 1995-02-14 US disclosed
WO-1994006757-A1 AGENTS ACTING AT CHOLECYSTOKININ RECEPTORS WARNER-LAMBERT COMPANY (US) 1994-03-31 WO disclosed