SCHEMBL8059348

SCHEMBL8059348

CC(C)c1[c]c(C(C)C)cc(-c2ccc3ccccc3n2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 14/20 0.49
NPC1 O15118 13/20 0.49
AR P10275 2/20 0.49
CYP3A4 P08684 2/20 0.49
CYP1A2 P05177 2/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
KDM4E B2RXH2 8/20 0.48
SMN1; SMN2 Q16637 8/20 0.48
ALDH1A1 P00352 8/20 0.48
NFKB1 P19838 2/20 0.47
NFKB2 Q00653 2/20 0.47
RELA Q04206 2/20 0.47
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
MAPT P10636 5/20 0.46
HSD17B10 Q99714 4/20 0.46
PKM P14618 4/20 0.46
HPGD P15428 4/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8043777 0.83 NPC1 (0.48) RAB9ANPC1ARCYP3A4CYP1A2
SCHEMBL25521681 0.76 AR (0.54) RAB9ANPC1ARCYP3A4CYP1A2
SCHEMBL1102504 0.75 RAB9A (0.66) RAB9ANPC1ARCYP3A4CYP1A2
SCHEMBL29638020 0.74 NPC1 (0.59) RAB9ANPC1ARCYP3A4CYP1A2
SCHEMBL10079213 0.74 NPC1 (0.59) RAB9ANPC1ARCYP3A4CYP1A2
SCHEMBL240431 0.73 NPC1 (0.63) RAB9ANPC1ARCYP3A4CYP1A2
SCHEMBL34467584 0.73 NPC1 (0.63) RAB9ANPC1ARCYP3A4CYP1A2
SCHEMBL21173048 0.73 RAB9A (0.60) RAB9ANPC1ARCYP3A4CYP1A2
SCHEMBL7005374 0.73 NPC1 (0.54) RAB9ANPC1ARCYP3A4CYP1A2
SCHEMBL4445443 0.73 NPC1 (0.47) RAB9ANPC1ARCYP3A4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001959-A1 METHOD FOR PRODUCING BIDENTATE MONOALKYL METAL COMPLEXES BASF AKTIENGESELLSCHAFT (DE) 2000-05-24 EP disclosed
WO-1999003867-A1 METHOD FOR PRODUCING BIDENTATE MONOALKYL METAL COMPLEXES BASF AKTIENGESELLSCHAFT (DE) 1999-01-28 WO disclosed