SCHEMBL8060293

SCHEMBL8060293

[O]CC[Si](c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.32

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
ALOX15 P16050 1/20 0.31
ALOX12 P18054 1/20 0.31
CASP1 P29466 1/20 0.31
HSD17B10 Q99714 1/20 0.31
ESR1 P03372 1/20 0.30
ESR2 Q92731 1/20 0.30
ADH1B P00325 1/20 0.30
ADH1C P00326 1/20 0.30
ADH1A P07327 1/20 0.30
ADH7 P40394 1/20 0.30
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10402043 0.83 CALM1 (0.35) MAPTALDH1A1ESR1ESR2
SCHEMBL3454933 0.75 MAPT (0.37) MAPTESR1ESR2
SCHEMBL4625996 0.74 ESR1 (0.30) ESR1ESR2
SCHEMBL23364946 0.74 ESR1 (0.30) ESR1ESR2
SCHEMBL28218923 0.74 TP53 (0.38) MAPTALDH1A1HPGDESR1ESR2
SCHEMBL23364915 0.74 ESR1 (0.30) ESR1ESR2
SCHEMBL23364934 0.74 ESR1 (0.30) ESR1ESR2
SCHEMBL4193671 0.74 IDO1 (0.38) ALDH1A1ESR1ESR2
SCHEMBL1043941 0.74 TDP1 (0.40) MAPTALDH1A1ESR1ESR2GAA
SCHEMBL7822716 0.73 KEAP1 (0.46) MAPTALDH1A1ESR1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4952690-A 6-substituted thia-aza compounds CIBA-GEIGY CORPORATION (US) 1990-08-28 US claimed
US-4447360-A Intermediates for thia-aza compounds with a β-lactam ring CIBA-GEIGY CORPORATION (US) 1984-05-08 US claimed
WO-2023223888-A1 METHOD FOR PRODUCING POLYCARBONATE RESIN, AND ALICYCLIC POLYCARBONATE RESIN 旭化成株式会社 2023-11-23 WO disclosed
WO-2023182378-A1 POLYCARBONATE RESIN, POLYCARBONATE RESIN COMPOSITION, OPTICAL COMPONENT, AND PRODUCTION METHOD FOR POLYCARBONATE RESIN 旭化成株式会社 2023-09-28 WO disclosed
US-20230192949-A1 POLYCARBONATE RESIN, POLYCARBONATE RESIN COMPOSITION, OPTICAL MOLDED ARTICLE COMPRISING SAME, AND CYCLIC CARBONATE ASAHI KASEI KABUSHIKI KAISHA (JP) 2023-06-22 US disclosed
EP-4092068-A1 POLYCARBONATE RESIN, POLYCARBONATE RESIN COMPOSITION, OPTICAL MOLDED BODY CONTAINING THESE, AND CYCLIC CARBONATE Asahi Kasei Kabushiki Kaisha (JP) 2022-11-23 EP disclosed
CN-114945619-A Polycarbonate resin, polycarbonate resin composition, optical molded article containing same, and cyclic carbonate 旭化成株式会社 2022-08-26 CN disclosed
WO-2021145443-A1 POLYCARBONATE RESIN, POLYCARBONATE RESIN COMPOSITION, OPTICAL MOLDED BODY CONTAINING THESE, AND CYCLIC CARBONATE 旭化成株式会社 2021-07-22 WO disclosed
US-6143724-A USED FOR TREATMENT, IMPROVEMENT AND PREVENTION OF INFLAMMATION AND DISEASES ACCOMPANYING INFLAMATION DAIKIN INDUSTRIES, LTD. (JP) 2000-11-07 US disclosed
EP-1013660-A1 2-FLUOROFUCOSYL-N-AROYLGLUCOSAMINE DERIVATIVES, INTERMEDIATES THEREFOR, AND PROCESSES FOR PRODUCING THESE Daikin Industries, Limited (JP) 2000-06-28 EP disclosed
EP-0832110-A1 ANTIVIRAL PEPTOID COMPOUNDS Novartis AG (CH) 1998-04-01 EP disclosed
WO-1996040759-A1 ANTIVIRAL PEPTOID COMPOUNDS NOVARTIS AG (CH) 1996-12-19 WO disclosed
US-4952690-A 6-substituted thia-aza compounds CIBA-GEIGY CORPORATION (US) 1990-08-28 US disclosed
US-4692442-A ANTIBIOTICS CIBA-GEIGY CORPORATION (US) 1987-09-08 US disclosed
US-4524028-A PENICILLINS CIBA-GEIGY CORPORATION (US) 1985-06-18 US disclosed
US-4518533-A Azetidinone-4-disulfides as intermediates for thia-aza compounds with a beta-lactam ring CIBA GEIGY CORPORATION (US) 1985-05-21 US disclosed
US-4515717-A INTERMEDIATES FOR 6-UNSUBSTITUTED PENICILLIN ANTIOBIOTICS CIBA GEIGY CORPORATION (US) 1985-05-07 US disclosed
US-4500457-A TREATING AN ACYLOXYAZETIDINONE WITH MERCAPTO COMPOUND, GLYOYLIC ESTER, HALOGENATION AGENT, AND PHOSPHINE COMPOUNT THEN CYCLIZATION CIBA-GEIGY CORPORATION (US) 1985-02-19 US disclosed
US-4447360-A Intermediates for thia-aza compounds with a β-lactam ring CIBA-GEIGY CORPORATION (US) 1984-05-08 US disclosed
US-4331676-A 2-PENEM COMPOUNDS UNSUBSTITUTED IN THE 6 POSITION CIBA-GEIGY CORPORATION (US) 1982-05-25 US disclosed