SCHEMBL8060520

SCHEMBL8060520

CCc1cc2c(cc1C(=O)OC)S(=O)(=O)CC(C)O2

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.35
TSHR P16473 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
ALDH1A1 P00352 8/20 0.34
HPGD P15428 3/20 0.34
GAA P10253 1/20 0.33
AKR1B1 P15121 1/20 0.33
KDM4E B2RXH2 4/20 0.33
MAOA P21397 1/20 0.32
SIRT1 Q96EB6 1/20 0.31
MAPT P10636 3/20 0.31
HSD17B10 Q99714 2/20 0.31
HTT P42858 1/20 0.31
REV1 Q9UBZ9 1/20 0.31
LMNA P02545 2/20 0.30
TP53 P04637 1/20 0.30
THRB P10828 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8058099 0.85 RAB9A (0.38) RAB9AMEN1KMT2AALDH1A1HPGD
SCHEMBL8045201 0.81 TSHR (0.34) RAB9ATSHRKMT2AALDH1A1HPGD
SCHEMBL8058197 0.80
SCHEMBL8060815 0.79 KDM4E (0.38) RAB9ATSHRMEN1KMT2AALDH1A1
SCHEMBL8062781 0.78 ALDH1A1 (0.36) TSHRKMT2AALDH1A1HPGDGAA
SCHEMBL8057027 0.78 RAB9A (0.43) RAB9AMEN1KMT2AALDH1A1HPGD
SCHEMBL8056335 0.77 ALDH1A1 (0.35) RAB9ATSHRALDH1A1HPGDKDM4E
SCHEMBL8056280 0.77 KDM4E (0.43) RAB9ATSHRMEN1KMT2AALDH1A1
SCHEMBL8062947 0.76 CA12 (0.36) RAB9ATSHRALDH1A1HPGDKDM4E
SCHEMBL8062773 0.75 TSHR (0.34) TSHRALDH1A1HPGDGAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed