SCHEMBL8056280

SCHEMBL8056280

CCc1cc2c(cc1C(=O)OC)S(=O)(=O)CCO2

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.43
ALDH1A1 P00352 6/20 0.43
MTNR1A P48039 1/20 0.40
GPR119 Q8TDV5 1/20 0.36
MAPT P10636 3/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
TP53 P04637 1/20 0.34
POLB P06746 1/20 0.34
HSD17B10 Q99714 3/20 0.34
RAB9A P51151 3/20 0.34
NPC1 O15118 2/20 0.33
TSHR P16473 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
RXFP1 Q9HBX9 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8060815 0.86 KDM4E (0.38) KDM4EALDH1A1GPR119MAPTSMN1; SMN2
SCHEMBL8056203 0.84 ALDH1A1 (0.44) KDM4EALDH1A1MTNR1AGPR119MAPT
SCHEMBL8057351 0.79
SCHEMBL8062947 0.78 CA12 (0.36) KDM4EALDH1A1MAPTSMN1; SMN2HSD17B10
SCHEMBL8060881 0.77 ALDH1A1 (0.35) KDM4EALDH1A1MAPTSMN1; SMN2KMT2A
SCHEMBL8062814 0.77 ALDH1A1 (0.35) KDM4EALDH1A1MAPTSMN1; SMN2KMT2A
SCHEMBL8045260 0.77 ALDH1A1 (0.33) KDM4EALDH1A1MAPTSMN1; SMN2KMT2A
SCHEMBL8060520 0.77 RAB9A (0.35) KDM4EALDH1A1MAPTKMT2AMEN1
SCHEMBL8060801 0.77 CTSL (0.34) KDM4EALDH1A1GPR119MAPTPOLB
SCHEMBL8060804 0.75 CYP2C9 (0.46) KDM4EALDH1A1MAPTSMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed