SCHEMBL8062828

SCHEMBL8062828

COC(=O)c1ccc2c(c1)S(=O)(=O)CCC2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA7 P43166 1/20 0.44
XDH P47989 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44
ALDH1A1 P00352 3/20 0.42
TRPA1 O75762 1/20 0.42
KDM4E B2RXH2 3/20 0.41
ATM Q13315 2/20 0.41
MAPT P10636 2/20 0.41
HPGD P15428 2/20 0.41
HSD17B10 Q99714 2/20 0.41
GLA P06280 1/20 0.41
GAA P10253 1/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
LMNA P02545 2/20 0.40
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8060786 0.91 CA1 (0.46) CA12CA1CA2CA7XDH
SCHEMBL26967607 0.84 GALR1 (0.48) CA12CA1CA2CA7CA9
SCHEMBL23705003 0.83 ALDH1A1 (0.56) CA12CA1CA2CA7CA9
SCHEMBL30058901 0.83 ALDH1A1 (0.56) CA12CA1CA2CA7CA9
SCHEMBL16212929 0.81 CA1 (0.43) CA1CA2CA9ALDH1A1LMNA
SCHEMBL8060691 0.79 LMNA (0.51) CA12CA1CA2CA7CA9
SCHEMBL7778601 0.78 CA2 (0.39) CA2LMNACYP2C9
SCHEMBL10502895 0.78 ATM (0.43) CA12CA1CA2CA7XDH
SCHEMBL21028293 0.78 CA1 (0.46) CA12CA1CA2CA7XDH
SCHEMBL23704889 0.78 ALDH1A1 (0.54) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed