SCHEMBL806308

SCHEMBL806308

C=C/C=C\C=C(/C)n1c(CSc2ncnc3nc[nH]c23)nc2ccsc2c1=O

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 4/20 0.59
ALDH1A1 P00352 1/20 0.46
HSD17B10 Q99714 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
PIK3CG P48736 9/20 0.43
POLB P06746 1/20 0.43
RECQL P46063 1/20 0.43
GAA P10253 1/20 0.41
PIK3CB P42338 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CDC7 O00311 4/20 0.40
DBF4 Q9UBU7 4/20 0.40
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL788778 0.74 PIK3CD (1.00) PIK3CDALDH1A1HSD17B10RXFP1PIK3CG
SCHEMBL1703918 0.62 PIK3CD (0.58) PIK3CDALDH1A1HSD17B10RXFP1PIK3CG
SCHEMBL16004753 0.59 PIK3CG (1.00) PIK3CDALDH1A1HSD17B10RXFP1PIK3CG
SCHEMBL10426489 0.59 G6PD (0.64) ALDH1A1HSD17B10CDC7DBF4TSHR
SCHEMBL31439407 0.57 PAK1 (0.71) ALDH1A1HSD17B10CDC7DBF4TSHR
SCHEMBL2115555 0.57 PAK1 (0.71) ALDH1A1HSD17B10CDC7DBF4TSHR
SCHEMBL29851680 0.57 CDC7 (1.00) ALDH1A1HSD17B10CDC7DBF4
SCHEMBL2120065 0.57 CDC7 (1.00) ALDH1A1HSD17B10CDC7DBF4
SCHEMBL3396404 0.57 TSHR (0.78) ALDH1A1POLBRECQLGAASMN1; SMN2
SCHEMBL10435363 0.56 CYP1A2 (1.00) ALDH1A1HSD17B10CDC7DBF4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037204-A1 INHIBITORS OF PI3K-DELTA AND METHODS OF THEIR USE AND MANUFACTURE EXELIXIS, INC. (US) 2012-03-22 WO disclosed