SCHEMBL8063808

SCHEMBL8063808

Cc1cc(C)cc(C(=O)CNC[C@@H](CC=O)c2ccc(Cl)c(Cl)c2)c1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HPGD P15428 1/20 0.35
S1PR2 O95136 2/20 0.34
S1PR4 O95977 2/20 0.34
S1PR3 Q99500 2/20 0.34
TACR1 P25103 2/20 0.34
S1PR1 P21453 1/20 0.34
ITGAV P06756 1/20 0.34
SLC6A2 P23975 4/20 0.33
SLC6A4 P31645 4/20 0.33
SLC6A3 Q01959 4/20 0.33
CYP3A4 P08684 3/20 0.33
CYP2D6 P10635 3/20 0.33
KCNH2 Q12809 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8053257 1.00 ALDH1A1 (0.37) ALDH1A1LMNAHTTSMN1; SMN2HPGD
SCHEMBL8580535 0.90 S1PR2 (0.43) ALDH1A1LMNAHTTSMN1; SMN2HPGD
SCHEMBL8069558 0.89 ALDH1A1 (0.38) ALDH1A1LMNAHTTSMN1; SMN2HPGD
SCHEMBL8069514 0.88 P2RY1 (0.36) ALDH1A1LMNAHTTSMN1; SMN2HPGD
SCHEMBL8561489 0.86 HTT (0.37) ALDH1A1LMNAHTTSMN1; SMN2HPGD
SCHEMBL8561494 0.86 HTT (0.37) ALDH1A1LMNAHTTSMN1; SMN2HPGD
SCHEMBL8064776 0.85 ALDH1A1 (0.36) ALDH1A1LMNAHTTSMN1; SMN2HPGD
SCHEMBL8064773 0.85 ALDH1A1 (0.36) ALDH1A1LMNAHTTSMN1; SMN2HPGD
SCHEMBL8560072 0.83 MCHR1 (0.39) ALDH1A1LMNAHTTSMN1; SMN2TACR1
SCHEMBL8560068 0.83 MCHR1 (0.39) ALDH1A1LMNAHTTSMN1; SMN2TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6013652-A ANTIINFLAMMATORY AGENTS; ANALGESICS; ANTIHISTAMINES MERCK & CO., INC. (US) 2000-01-11 US disclosed
US-5962462-A COMPOUNDS WHICH INHIBIT THE ENTRY OF HUMAN IMMUNODEFICIENCY VIRUS (HIV) INTO TARGET CELLS; DELAYING THE ONSET OF ACQUIRED IMMUNE DEFICIENCY SYNDROME (AIDS). MERCK & CO., INC. (US) 1999-10-05 US disclosed
WO-1998025605-A1 SPIRO-SUBSTITUTED AZACYCLES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO., INC. (US) 1998-06-18 WO disclosed
EP-0702681-A1 SPIRO-SUBSTITUTED AZACYCLES AS NEUROKININ ANTAGONISTS MERCK & CO. INC. (US) 1996-03-27 EP disclosed
WO-1994029309-A1 SPIRO-SUBSTITUTED AZACYCLES AS NEUROKININ ANTAGONISTS MERCK & CO., INC. (US) 1994-12-22 WO disclosed