SCHEMBL8580535

SCHEMBL8580535

Cc1cccc(C(=O)CNCC(CC=O)c2ccc(Cl)c(Cl)c2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR2 O95136 1/20 0.43
S1PR4 O95977 1/20 0.43
S1PR3 Q99500 1/20 0.43
MEN1 O00255 2/20 0.39
MAPT P10636 2/20 0.39
KMT2A Q03164 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
LMNA P02545 2/20 0.39
HTT P42858 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39
MCHR1 Q99705 1/20 0.37
NLRP3 Q96P20 1/20 0.36
ATM Q13315 1/20 0.36
ALDH1A1 P00352 3/20 0.35
TDP2 O95551 1/20 0.35
ALDH3A1 P30838 1/20 0.35
GPR139 Q6DWJ6 1/20 0.35
HDAC8 Q9BY41 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8063808 0.90 ALDH1A1 (0.37) S1PR2S1PR4S1PR3LMNAHTT
SCHEMBL8053257 0.90 ALDH1A1 (0.37) S1PR2S1PR4S1PR3LMNAHTT
SCHEMBL8069514 0.83 P2RY1 (0.36) S1PR4S1PR3LMNAHTTSMN1; SMN2
SCHEMBL8069558 0.79 ALDH1A1 (0.38) S1PR2S1PR4S1PR3MAPTKMT2A
SCHEMBL8560068 0.78 MCHR1 (0.39) MEN1KMT2ALMNAHTTSMN1; SMN2
SCHEMBL8560072 0.78 MCHR1 (0.39) MEN1KMT2ALMNAHTTSMN1; SMN2
SCHEMBL8580532 0.78 TACR2 (0.51)
SCHEMBL8561489 0.76 HTT (0.37) S1PR2S1PR4S1PR3LMNAHTT
SCHEMBL8561494 0.76 HTT (0.37) S1PR2S1PR4S1PR3LMNAHTT
SCHEMBL8064776 0.76 ALDH1A1 (0.36) S1PR2S1PR4S1PR3LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998025617-A1 SUBSTITUTED ARYL PIPERAZINES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO., INC. (US) 1998-06-18 WO disclosed
US-5607936-A USEFUL IN TREATMENT OF RESPIRATORY DISEASES MERCK & CO., INC. (US) 1997-03-04 US disclosed