SCHEMBL8064901

SCHEMBL8064901

CCc1ccc(C(O)c2cccc(F)c2)cc1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
ATM Q13315 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
BRD4 O60885 2/20 0.41
CREBBP Q92793 1/20 0.41
SLC6A2 P23975 2/20 0.40
SLC6A4 P31645 2/20 0.40
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
CNR2 P34972 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8064702 0.87 KMT2A (0.40) CES2CES1BRD4CREBBPSLC6A2
SCHEMBL8064208 0.82 LMNA (0.53) TSHRMAPK1ATMTDP1L3MBTL1
SCHEMBL230519 0.82 CES2 (0.49) CES2CES1BRD4HDAC4HDAC7
SCHEMBL8077592 0.82 CES2 (0.44) L3MBTL1CES2CES1BRD4CREBBP
SCHEMBL227352 0.82 CES2 (0.55) CES2CES1BRD4SLC6A2SLC6A4
SCHEMBL28788047 0.81 BRD4 (0.49) CES2CES1BRD4CREBBPSLC6A2
SCHEMBL1632280 0.80 TSHR (0.42) TSHRMAPK1ATMTDP1L3MBTL1
SCHEMBL230487 0.80 IDO1 (0.52) CES2CES1BRD4SLC6A2SLC6A4
SCHEMBL6899388 0.80 TP53 (0.54) TSHRMAPK1ATMTDP1L3MBTL1
SCHEMBL6349980 0.77 CES2 (0.45) CES2CES1BRD4SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6166072-A Amino acid derivatives ALLELIX NEUROSCIENCE, INC. (CA) 2000-12-26 US disclosed
WO-1999034790-A1 GLYCINE TRANSPORT INHIBITORS ALLELIX NEUROSCIENCE, INC. (US) 1999-07-15 WO disclosed