SCHEMBL8065484

SCHEMBL8065484

Cc1c(N)ccc(Cc2ccc(N)c(C)c2N)c1N

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.42
TSHR P16473 4/20 0.42
PIK3CA P42336 1/20 0.42
ALDH1A1 P00352 8/20 0.39
ALOX15 P16050 3/20 0.39
HSD17B10 Q99714 2/20 0.39
CYP1A2 P05177 1/20 0.39
CASP7 P55210 1/20 0.39
HIF1A Q16665 1/20 0.39
TDP1 Q9NUW8 4/20 0.39
TP53 P04637 2/20 0.39
THRB P10828 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
MAPK1 P28482 1/20 0.34
HTT P42858 1/20 0.34
POLB P06746 1/20 0.32
CD44 P16070 1/20 0.32
SLC6A2 P23975 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8063101 0.83 CYP3A4 (0.48) CYP3A4TSHRALDH1A1CYP1A2TDP1
SCHEMBL10845366 0.83 HTR2A (0.41) CYP3A4TSHRPIK3CAALDH1A1ALOX15
SCHEMBL2776271 0.83 ALDH1A1 (0.40) CYP3A4TSHRPIK3CAALDH1A1ALOX15
SCHEMBL39192 0.82 CYP3A4 (0.43) CYP3A4TSHRPIK3CAALDH1A1ALOX15
SCHEMBL8538345 0.81 CYP3A4 (0.39) CYP3A4TSHRPIK3CAALDH1A1ALOX15
SCHEMBL17998039 0.81 CYP3A4 (0.39) CYP3A4TSHRPIK3CAALDH1A1ALOX15
SCHEMBL11466097 0.80 SKP2 (0.47) CYP3A4TSHRALDH1A1ALOX15HSD17B10
SCHEMBL30906995 0.80 SKP2 (0.47) CYP3A4TSHRALDH1A1ALOX15HSD17B10
SCHEMBL6320495 0.80 POLB (0.42) CYP3A4TSHRPIK3CAALDH1A1ALOX15
SCHEMBL3674174 0.78 GABRA1 (0.36) TSHRALDH1A1ALOX15HSD17B10CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0668101-B1 Ruthenium catalysts, their preparation and their use in the preparation of cycloaliphatic polyamines BAYER AG (DE) 2000-06-07 EP disclosed
US-5663443-A HYDROGENATION BAYER AKTIENGESELLSCHAFT (DE) 1997-09-02 US disclosed
EP-0668101-A1 Ruthenium catalysts, their preparation and their use in the preparation of cycloaliphatic polyamines BAYER AG (DE) 1995-08-23 EP disclosed