SCHEMBL8066780

SCHEMBL8066780

NC(=O)c1cc([N+](=O)[O-])c(Cl)c([N+](=O)[O-])c1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C19 P33261 1/20 0.48
LMNA P02545 2/20 0.46
KMT2A Q03164 1/20 0.46
TSHR P16473 3/20 0.46
GPR35 Q9HC97 1/20 0.44
CYP3A4 P08684 4/20 0.43
MAPT P10636 1/20 0.43
BLM P54132 1/20 0.43
PMP22 Q01453 1/20 0.43
PARP1 P09874 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
CASP1 P29466 1/20 0.41
VCAM1 P19320 2/20 0.40
HPGD P15428 1/20 0.40
ALOX15 P16050 1/20 0.40
HIF1A Q16665 1/20 0.40
TXNRD1 Q16881 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11317490 0.85 LMNA (0.44) ALDH1A1CYP1A2CYP2D6CYP2C19LMNA
SCHEMBL3291904 0.84 ALDH1A1 (0.60) ALDH1A1CYP1A2CYP2D6CYP2C19LMNA
SCHEMBL1478701 0.84 ALDH1A1 (0.60) ALDH1A1CYP1A2CYP2D6CYP2C19LMNA
SCHEMBL10558853 0.84 TSHR (0.47) ALDH1A1CYP1A2CYP2D6CYP2C19TSHR
SCHEMBL9899863 0.81 ALDH1A1 (0.47) ALDH1A1CYP1A2CYP2D6CYP2C19LMNA
SCHEMBL9859808 0.81 ALDH1A1 (0.49) ALDH1A1LMNAKMT2ATSHRGPR35
SCHEMBL6121980 0.81 ALDH1A1 (0.47) ALDH1A1LMNAKMT2ATSHRGPR35
SCHEMBL2889129 0.79 ALDH1A1 (0.68) ALDH1A1CYP1A2LMNAKMT2ATSHR
SCHEMBL7644871 0.79 TSHR (0.62) ALDH1A1CYP1A2CYP2D6CYP2C19KMT2A
SCHEMBL8064653 0.79 PDGFRB (0.48) ALDH1A1CYP1A2CYP2D6CYP2C19LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1016405-A2 Arylating medicaments Radopath Pharmaceuticals International Limited (GB) 2000-07-05 EP claimed
CN-1124012-A Arylating medicaments RADOPATH LTD (GB) 1996-06-05 CN claimed
EP-0700287-A1 ARYLATING MEDICAMENTS RADOPATH LIMITED (GB) 1996-03-13 EP claimed
WO-1994027584-A2 ARYLATING MEDICAMENTS RADOPATH LIMITED (GB) 1994-12-08 WO claimed
EP-1016405-A2 Arylating medicaments Radopath Pharmaceuticals International Limited (GB) 2000-07-05 EP disclosed
EP-0700287-A1 ARYLATING MEDICAMENTS RADOPATH LIMITED (GB) 1996-03-13 EP disclosed
WO-1994027584-A2 ARYLATING MEDICAMENTS RADOPATH LIMITED (GB) 1994-12-08 WO disclosed
US-4169153-A PROPHYLAXIS, ANTIHISTAMINES THE UPJOHN COMPANY (US) 1979-09-25 US disclosed
US-4091011-A PROPHYLACTIC ANTIANAPHYLACTICS, ANTIALLERGENS THE UPJOHN COMPANY (US) 1978-05-23 US disclosed