SCHEMBL8066880

SCHEMBL8066880

CCOc1cccc(CNC(=O)c2cc(-c3nn[nH]n3)cc(C)n2)c1

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
XDH P47989 2/20 0.56
MMP13 P45452 16/20 0.53
ROCK2 O75116 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
ROCK1 Q13464 1/20 0.52
MMP3 P08254 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3688685 0.90 MMP13 (0.63) MMP13ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL8072658 0.90 MMP13 (0.53) XDHMMP13ROCK2CYP3A4CYP2D6
SCHEMBL8057403 0.80 MMP13 (0.62) MMP13ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL8058261 0.80 MMP13 (0.51) XDHMMP13ROCK2CYP3A4CYP2D6
SCHEMBL4182437 0.79 MMP13 (0.61) XDHMMP13
SCHEMBL8056592 0.79 MMP13 (0.59) MMP13
SCHEMBL3694242 0.77 MMP13 (0.62) MMP13ROCK2ROCK1
SCHEMBL8070170 0.77 MMP13 (0.61) MMP13
SCHEMBL8070443 0.77 MMP13 (0.85) MMP13MMP3
SCHEMBL8059690 0.77 MMP13 (0.85) MMP13MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009016498-A1 PYRIMIDINE AND PYRIDINE DERIVATIVES AND THEIR PHARMACEUTICAL USE AND COMPOSITIONS PFIZER INC. (US) 2009-02-05 WO disclosed