SCHEMBL8058261

SCHEMBL8058261

Cc1nc(C(=O)NCc2cccc(OCCO)c2)cc(-c2nn[nH]n2)n1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 7/20 0.51
ROCK2 O75116 3/20 0.45
CYP3A4 P08684 3/20 0.45
CYP2D6 P10635 3/20 0.45
CYP2C9 P11712 3/20 0.45
ROCK1 Q13464 3/20 0.45
AGTR1 P30556 2/20 0.44
XDH P47989 1/20 0.43
MMP3 P08254 1/20 0.42
MAPT P10636 1/20 0.42
ADORA3 P0DMS8 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA2B P29275 1/20 0.41
ADORA1 P30542 1/20 0.41
EDNRA P25101 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3765203 0.90 MMP13 (0.57) MMP13ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL8071850 0.84 MMP13 (0.52) MMP13ROCK2ROCK1AGTR1XDH
SCHEMBL8072658 0.81 MMP13 (0.53) MMP13ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL8066880 0.80 XDH (0.56) MMP13ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL8071844 0.80 ROCK1 (0.49) MMP13ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL8055185 0.78 MMP13 (0.54) MMP13XDHADORA2AADORA1
SCHEMBL3688685 0.77 MMP13 (0.63) MMP13ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL8070937 0.77 MMP13 (0.57) MMP13ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL3686913 0.77 MMP13 (0.58) MMP13ROCK2ROCK1AGTR1
SCHEMBL3690556 0.77 MMP13 (0.44) MMP13AGTR1XDHADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009016498-A1 PYRIMIDINE AND PYRIDINE DERIVATIVES AND THEIR PHARMACEUTICAL USE AND COMPOSITIONS PFIZER INC. (US) 2009-02-05 WO disclosed