SCHEMBL8068291

SCHEMBL8068291

CC1(C)OCC(CON2c3nc[nH]c3C(=O)NC2N)O1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.37
ALDH1A1 P00352 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36
CCNK O75909 1/20 0.33
CDK12 Q9NYV4 1/20 0.33
KCNJ5 P48544 2/20 0.31
KCNJ3 P48549 2/20 0.31
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
TP53 P04637 1/20 0.31
CYP3A4 P08684 1/20 0.31
MAPT P10636 1/20 0.31
PKM P14618 1/20 0.31
HPGD P15428 1/20 0.31
ALOX15 P16050 1/20 0.31
MAPK1 P28482 1/20 0.31
CASP1 P29466 1/20 0.31
BLM P54132 1/20 0.31
KMT2A Q03164 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6263155 0.67 CA2 (0.37) CA2ALDH1A1NPSR1CCNKCDK12
SCHEMBL6035382 0.65 GDA (0.35)
SCHEMBL6845476 0.61 ALDH1A1 (0.45) CA2ALDH1A1NPSR1KDM4EMEN1
SCHEMBL4860312 0.61 ALDH1A1 (0.45) CA2ALDH1A1NPSR1KDM4EMEN1
SCHEMBL4860306 0.61 ALDH1A1 (0.45) CA2ALDH1A1NPSR1KDM4EMEN1
SCHEMBL30486880 0.61 ALDH1A1 (0.45) CA2ALDH1A1NPSR1KDM4EMEN1
SCHEMBL4428837 0.60 CDK1 (0.57)
SCHEMBL7981045 0.60 CDK1 (0.57)
SCHEMBL21911823 0.60 TMEM97 (0.39) CA2ALDH1A1NPSR1KDM4EMEN1
SCHEMBL10471467 0.59 CCNK (0.39) CA2ALDH1A1NPSR1CCNKCDK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1017394-A1 CYCLIN DEPENDENT KINASE INHIBITING PURINE DERIVATIVES CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 2000-07-12 EP disclosed
WO-1999002162-A9 CYCLIN DEPENDENT KINASE INHIBITING PURINE DERIVATIVES CANCER RES CAMPAIGN TECH (GB) 1999-07-29 WO disclosed
WO-1999002162-A1 CYCLIN DEPENDENT KINASE INHIBITING PURINE DERIVATIVES CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 1999-01-21 WO disclosed