SCHEMBL8068331

SCHEMBL8068331

COc1cc(CNC(=O)c2cc(-c3nc[nH]n3)cc(C)n2)ccc1F

nearest known ligand 0.60

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 16/20 0.60
ROCK2 O75116 1/20 0.50
ROCK1 Q13464 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8068866 0.89 MMP13 (0.57) MMP13
SCHEMBL3694242 0.88 MMP13 (0.62) MMP13ROCK2ROCK1
SCHEMBL8069461 0.86 MMP13 (0.58) MMP13ROCK2ROCK1
SCHEMBL8057403 0.82 MMP13 (0.62) MMP13ROCK2ROCK1
SCHEMBL8071335 0.81 MMP13 (0.58) MMP13ROCK2ROCK1
SCHEMBL8066239 0.79 MMP13 (0.72) MMP13
SCHEMBL8056484 0.79 MMP13 (0.53) MMP13ROCK2ROCK1
SCHEMBL8068867 0.78 MMP13 (0.72) MMP13
SCHEMBL8069587 0.78 MMP13 (0.72) MMP13
SCHEMBL8065705 0.77 MMP13 (0.87) MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101815710-A Pyrimidine and pyridine derivatives, their pharmaceutical use and compositions PFIZER 2010-08-25 CN disclosed
WO-2009016498-A1 PYRIMIDINE AND PYRIDINE DERIVATIVES AND THEIR PHARMACEUTICAL USE AND COMPOSITIONS PFIZER INC. (US) 2009-02-05 WO disclosed