SCHEMBL8069461

SCHEMBL8069461

COc1cc(CNC(=O)c2cc(-c3nc[nH]n3)nc(C)n2)ccc1F

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 8/20 0.58
ROCK2 O75116 2/20 0.47
ROCK1 Q13464 2/20 0.47
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
NOD2 Q9HC29 1/20 0.44
L3MBTL1 Q9Y468 2/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPK1 P28482 1/20 0.42
HTT P42858 1/20 0.42
ADORA2A P29274 1/20 0.41
ADORA1 P30542 1/20 0.41
MMP10 P09238 1/20 0.40
MMP9 P14780 1/20 0.40
MMP8 P22894 1/20 0.40
PDE2A O00408 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8056484 0.91 MMP13 (0.53) MMP13ROCK2ROCK1MEN1KMT2A
SCHEMBL3686913 0.86 MMP13 (0.58) MMP13ROCK2ROCK1MEN1KMT2A
SCHEMBL8068331 0.86 MMP13 (0.60) MMP13ROCK2ROCK1
SCHEMBL8070937 0.83 MMP13 (0.57) MMP13ROCK2ROCK1MEN1KMT2A
SCHEMBL8065850 0.81 MMP13 (0.53) MMP13ROCK2ROCK1MEN1KMT2A
SCHEMBL3762298 0.81 MMP13 (0.53) MMP13ROCK2ROCK1MEN1KMT2A
SCHEMBL13729454 0.81 MMP13 (0.53) MMP13ROCK2ROCK1MEN1KMT2A
SCHEMBL13728389 0.80 MMP13 (0.55) MMP13ROCK2ROCK1MEN1KMT2A
SCHEMBL8068341 0.80 MMP13 (0.52) MMP13ROCK2ROCK1MEN1KMT2A
SCHEMBL8067164 0.80 MMP13 (0.54) MMP13ROCK2ROCK1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009016498-A1 PYRIMIDINE AND PYRIDINE DERIVATIVES AND THEIR PHARMACEUTICAL USE AND COMPOSITIONS PFIZER INC. (US) 2009-02-05 WO disclosed