SCHEMBL8069879

SCHEMBL8069879

CC(C)[C@H](N)C(=O)N[C@H](C)c1nc2ccccc2s1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.52
ALOX15 P16050 1/20 0.49
TSHR P16473 1/20 0.49
CASP1 P29466 1/20 0.49
LOXL2 Q9Y4K0 1/20 0.49
RAB9A P51151 2/20 0.47
HPGD P15428 2/20 0.47
ALDH1A1 P00352 2/20 0.47
NPC1 O15118 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
HIF1A Q16665 1/20 0.47
HSD17B10 Q99714 1/20 0.47
FFAR2 O15552 1/20 0.43
ADORA1 P30542 1/20 0.43
DYRK1A Q13627 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8069848 0.82 PPARA (0.46) ALOX5
SCHEMBL8060776 0.78 TSHR (0.46) ALOX5ALOX15TSHRCASP1RAB9A
SCHEMBL8060795 0.78 TSHR (0.46) ALOX5ALOX15TSHRCASP1RAB9A
SCHEMBL8060765 0.77 HDAC3 (0.46) ALOX15TSHRCASP1HPGDALDH1A1
SCHEMBL8069877 0.76 ALOX5 (0.55) ALOX5ALOX15TSHRCASP1LOXL2
SCHEMBL10480454 0.75 LOXL2 (0.57) ALOX5ALOX15TSHRCASP1LOXL2
SCHEMBL8895495 0.75 ALOX5 (0.51) ALOX5ALOX15CYP1A2
SCHEMBL2839532 0.74 LOXL2 (0.64) ALOX5ALOX15TSHRCASP1LOXL2
SCHEMBL8175754 0.74 ALOX5 (0.49) ALOX5ALOX15TSHRCASP1LOXL2
SCHEMBL7285854 0.73 ALOX15 (0.58) ALOX5ALOX15TSHRCASP1LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0775696-B1 AMINO ACID AMIDE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AGROHORTICULTURAL FUNGICIDE, AND FUNGICIDAL METHOD KUMIAI CHEMICAL INDUSTRY CO (JP) 2000-07-19 EP disclosed
EP-0775696-A1 AMINO ACID AMIDE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AGROHORTICULTURAL FUNGICIDE, AND FUNGICIDAL METHOD KumaiI Chemical Industry Co., Ltd. (JP) 1997-05-28 EP disclosed