SCHEMBL8070147

SCHEMBL8070147

N=C(N)NC(=O)c1ccc(Oc2ccc(S(N)(=O)=O)cc2)c(C(F)(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.40
CA2 P00918 4/20 0.39
CA1 P00915 3/20 0.39
CA9 Q16790 3/20 0.39
CA7 P43166 2/20 0.39
ALDH1A1 P00352 2/20 0.39
KMT2A Q03164 1/20 0.39
HTT P42858 1/20 0.38
KIF11 P52732 1/20 0.38
CCR2 P41597 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8059411 0.93 HDAC3 (0.39) CCR2
SCHEMBL8061430 0.89 MRGPRX1 (0.40) CCR2
SCHEMBL8767698 0.86 F2 (0.45)
Hydrochloric Acid SCHEMBL8505884 0.85 F2 (0.44)
Hydrochloric Acid SCHEMBL8506593 0.84 BRAF (0.43) KMT2ACCR2
Hydrochloric Acid SCHEMBL8503960 0.84 STK39 (0.45)
SCHEMBL8445993 0.83 ALDH1A1 (0.48) ALDH1A1KMT2A
SCHEMBL8059621 0.82 SLC6A4 (0.43) TSHRALDH1A1KMT2AHTTCCR2
Hydrochloric Acid SCHEMBL8070562 0.82 ALDH1A1 (0.47) ALDH1A1KMT2A
SCHEMBL8075090 0.82 CA1 (0.52) CA2CA1CA9ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057322-A USEFUL IN TREATMENT OF CARDIOVASCULAR DISEASES HOECHST AKTIENGESELLSCHAFT (DE) 2000-05-02 US disclosed
EP-0723956-B1 Basically substituted benzoylguanidines, process for their preparation, their use as medicaments or diagnostics as well as medicaments containing them HOECHST AG (DE) 1999-10-13 EP disclosed
EP-0723956-A1 Basically substituted benzoylguanidines, process for their preparation, their use as medicaments or diagnostics as well as medicaments containing them HOECHST AKTIENGESELLSCHAFT (DE) 1996-07-31 EP disclosed