SCHEMBL8070663

SCHEMBL8070663

COc1cc(CNC(=O)c2cc(-c3ncn(C[C@H]4CC[C@H](NC(=O)OC(C)(C)C)CC4)n3)nc(C)n2)ccc1F

nearest known ligand 0.53

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 16/20 0.53
NAMPT P43490 1/20 0.37
MCHR1 Q99705 1/20 0.36
DRD2 P14416 1/20 0.36
ROCK2 O75116 1/20 0.36
ROCK1 Q13464 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8072927 0.93 MMP13 (0.49) MMP13NAMPT
SCHEMBL3808479 0.92 MMP13 (0.56) MMP13MCHR1
SCHEMBL3808476 0.92 MMP13 (0.56) MMP13MCHR1
SCHEMBL8069457 0.91 MMP13 (0.54) MMP13
SCHEMBL8071946 0.90 MMP13 (0.55) MMP13MCHR1
SCHEMBL8068891 0.89 MMP13 (0.61) MMP13
SCHEMBL3805240 0.88 MMP13 (0.67) MMP13
SCHEMBL3805239 0.88 MMP13 (0.67) MMP13
SCHEMBL8065798 0.88 MMP13 (0.53) MMP13ROCK2ROCK1
SCHEMBL8074480 0.88 MMP13 (0.56) MMP13ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009016498-A1 PYRIMIDINE AND PYRIDINE DERIVATIVES AND THEIR PHARMACEUTICAL USE AND COMPOSITIONS PFIZER INC. (US) 2009-02-05 WO disclosed