SCHEMBL8071748

SCHEMBL8071748

COc1cc2nc(N3CCC(Nc4ccc(C(=O)O)cn4)CC3)nc(N)c2cc1OC

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 3/20 0.60
ADRA1B P35368 3/20 0.60
KDM4E B2RXH2 3/20 0.55
ALDH1A1 P00352 3/20 0.55
HPGD P15428 3/20 0.55
GLA P06280 2/20 0.55
HSD17B10 Q99714 2/20 0.55
ADRA1D P25100 2/20 0.55
TP53 P04637 1/20 0.55
TSHR P16473 1/20 0.55
MAPK1 P28482 1/20 0.55
SLC22A1 O15245 1/20 0.55
ABCC4 O15439 1/20 0.55
LMNA P02545 1/20 0.55
ADRA2A P08913 1/20 0.55
GAA P10253 1/20 0.55
ADRA2B P18089 1/20 0.55
ADRA2C P18825 1/20 0.55
DRD1 P21728 1/20 0.55
ACHE P22303 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8071651 0.93 ADRA1A (0.57) ADRA1AADRA1BKDM4EALDH1A1HPGD
SCHEMBL8071911 0.88 ADRA1A (0.62) ADRA1AADRA1B
SCHEMBL8071831 0.85 KDM4E (0.55) ADRA1AADRA1BKDM4EALDH1A1HPGD
SCHEMBL8077026 0.82 ADRA1A (0.60) ADRA1AADRA1BADRA1DADRA2AADRA2B
SCHEMBL8077031 0.82 KDM4E (0.55) ADRA1AADRA1BKDM4EALDH1A1HPGD
SCHEMBL8071975 0.82 ADRA1A (0.56) ADRA1AADRA1B
SCHEMBL8076826 0.79 ADRA1A (0.56) ADRA1AADRA1BADRA1D
SCHEMBL8075296 0.78 EHMT2 (0.55) ADRA1AADRA1BKDM4EALDH1A1HPGD
SCHEMBL8070244 0.77 EHMT2 (0.52) ADRA1AADRA1B
SCHEMBL11398578 0.77 KDM4E (0.65) KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6156758-A Antibacterial quinazoline compounds ISIS PHARMACEUTICALS, INC. (US) 2000-12-05 US disclosed