SCHEMBL8071790

SCHEMBL8071790

CCC(Br)C(=O)c1ccc(S(C)(=O)=O)cc1

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GSR P00390 2/20 0.46
PTGS2 P35354 2/20 0.45
ENPP2 Q13822 1/20 0.44
AKR1C3 P42330 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18193727 0.86 GSR (0.44) GSRPTGS2ENPP2AKR1C3
SCHEMBL28427675 0.83 GSK3B (0.53) GSRPTGS2ENPP2AKR1C3
SCHEMBL7481806 0.81 ENPP2 (0.47) GSRPTGS2ENPP2AKR1C3
SCHEMBL5502450 0.80 TDP1 (0.46) AKR1C3
SCHEMBL3110619 0.79 GSK3B (0.48)
SCHEMBL3033043 0.79 SLC6A2 (0.47)
SCHEMBL11835508 0.78 HPGD (0.56) PTGS2
SCHEMBL7878318 0.78 HTT (0.51)
SCHEMBL2702007 0.78 PTPN1 (0.47)
SCHEMBL4421773 0.78 LMNA (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1023277-A1 NOVEL 3,4-DIARYLTHIAZOLIN-2-ONE OR -2-THIONE DERIVATIVES, PREPARATION METHODS AND USES IN THERAPY LABORATOIRES UPSA (FR) 2000-08-02 EP disclosed
WO-1999018093-A1 NOVEL 3,4-DIARYLTHIAZOLIN-2-ONE OR -2-THIONE DERIVATIVES, PREPARATION METHODS AND USES IN THERAPY LABORATOIRES UPSA (FR) 1999-04-15 WO disclosed