SCHEMBL28427675

SCHEMBL28427675

CS(=O)(=O)c1ccc(C(=O)C(Br)Br)cc1

nearest known ligand 0.56

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 3/20 0.53
ENPP2 Q13822 2/20 0.48
AKR1C3 P42330 3/20 0.46
GSR P00390 2/20 0.46
PTGS2 P35354 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7481806 0.86 ENPP2 (0.47) ENPP2AKR1C3GSRPTGS2
SCHEMBL8071790 0.83 GSR (0.46) ENPP2AKR1C3GSRPTGS2
SCHEMBL10747959 0.82 ENPP2 (0.42) ENPP2AKR1C3GSRPTGS2
SCHEMBL8049079 0.82 ENPP2 (0.50) ENPP2AKR1C3GSRPTGS2
SCHEMBL18193727 0.80 GSR (0.44) ENPP2AKR1C3GSRPTGS2
SCHEMBL8722500 0.80 ENPP2 (0.48) ENPP2AKR1C3GSRPTGS2
SCHEMBL9644843 0.80 GSK3B (0.76) GSK3B
SCHEMBL7836035 0.79 PTGS2 (0.49) AKR1C3PTGS2
SCHEMBL7084244 0.77 EPHX2 (0.53) AKR1C3PTGS2
SCHEMBL8562014 0.77 EPHX2 (0.53) AKR1C3PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108864003-B Preparation method of dapoxib intermediate and dapoxib 江苏美迪克化学品有限公司 2020-06-16 CN claimed
CN-108864003-B Preparation method of dapoxib intermediate and dapoxib 江苏美迪克化学品有限公司 2020-06-16 CN disclosed
CN-108864003-B Preparation method of dapoxib intermediate and dapoxib 江苏美迪克化学品有限公司 2020-06-16 CN disclosed