SCHEMBL8071850

SCHEMBL8071850

Cc1nc(C(=O)NCc2ccc(F)c(OCCO)c2)cc(-c2nn[nH]n2)n1

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 11/20 0.52
XDH P47989 1/20 0.42
KDM4C Q9H3R0 1/20 0.40
EPHX2 P34913 1/20 0.40
NR1H4 Q96RI1 1/20 0.40
CTSD P07339 3/20 0.40
AGTR1 P30556 1/20 0.39
ROCK2 O75116 1/20 0.39
ROCK1 Q13464 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3686913 0.90 MMP13 (0.58) MMP13CTSDAGTR1ROCK2ROCK1
SCHEMBL8056484 0.88 MMP13 (0.53) MMP13ROCK2ROCK1
SCHEMBL8055185 0.86 MMP13 (0.54) MMP13XDHKDM4CEPHX2NR1H4
SCHEMBL3690556 0.84 MMP13 (0.44) MMP13XDHKDM4CEPHX2NR1H4
SCHEMBL3696323 0.84 MMP13 (0.44) MMP13XDHKDM4CEPHX2NR1H4
SCHEMBL8069852 0.84 MMP13 (0.47) MMP13XDHKDM4CEPHX2NR1H4
SCHEMBL8058261 0.84 MMP13 (0.51) MMP13XDHAGTR1ROCK2ROCK1
SCHEMBL8055078 0.80 MMP13 (0.47) MMP13ROCK2ROCK1
SCHEMBL8066347 0.79 MMP13 (0.47) MMP13ROCK2ROCK1
SCHEMBL8065771 0.78 MMP13 (0.51) MMP13XDHCTSDROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009016498-A1 PYRIMIDINE AND PYRIDINE DERIVATIVES AND THEIR PHARMACEUTICAL USE AND COMPOSITIONS PFIZER INC. (US) 2009-02-05 WO disclosed