SCHEMBL8069852

SCHEMBL8069852

Cc1nc(C(=O)NCc2ccc(F)c(Cl)c2)cc(-c2nn[nH]n2)n1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 7/20 0.47
HDAC3 O15379 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
WDR5 P61964 3/20 0.41
EPHX2 P34913 1/20 0.41
NR1H4 Q96RI1 1/20 0.41
MAPK1 P28482 3/20 0.40
KDM4C Q9H3R0 1/20 0.39
PTGER4 P35408 1/20 0.39
XDH P47989 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8055185 0.90 MMP13 (0.54) MMP13EPHX2NR1H4KDM4CXDH
SCHEMBL3696323 0.89 MMP13 (0.44) MMP13EPHX2NR1H4KDM4CXDH
SCHEMBL3690556 0.89 MMP13 (0.44) MMP13EPHX2NR1H4KDM4CXDH
SCHEMBL3686913 0.87 MMP13 (0.58) MMP13
SCHEMBL8070170 0.85 MMP13 (0.61) MMP13EPHX2NR1H4
SCHEMBL8071850 0.84 MMP13 (0.52) MMP13EPHX2NR1H4KDM4CXDH
SCHEMBL8061043 0.84 MMP13 (0.51) MMP13HDAC3HDAC1HDAC2HDAC6
SCHEMBL3765203 0.79 MMP13 (0.57) MMP13
SCHEMBL8058261 0.77 MMP13 (0.51) MMP13XDH
SCHEMBL8056592 0.75 MMP13 (0.59) MMP13EPHX2NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009016498-A1 PYRIMIDINE AND PYRIDINE DERIVATIVES AND THEIR PHARMACEUTICAL USE AND COMPOSITIONS PFIZER INC. (US) 2009-02-05 WO disclosed