SCHEMBL8072341

SCHEMBL8072341

COc1cccc(CNC(=O)c2cc(C(N)=O)cc(C)n2)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 12/20 0.59
ADORA3 P0DMS8 1/20 0.57
ADORA2A P29274 1/20 0.57
ADORA2B P29275 1/20 0.57
ADORA1 P30542 1/20 0.57
MMP3 P08254 1/20 0.56
CHRM4 P08173 1/20 0.56
HPGD P15428 2/20 0.54
KDM4E B2RXH2 2/20 0.54
USP2 O75604 1/20 0.54
ALDH1A1 P00352 1/20 0.54
LMNA P02545 1/20 0.54
ROCK2 O75116 1/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2D6 P10635 1/20 0.54
CYP2C9 P11712 1/20 0.54
PRKACA P17612 1/20 0.54
GSK3A P49840 1/20 0.54
GSK3B P49841 1/20 0.54
PRKX P51817 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8062920 0.85 CHRM4 (0.51) MMP13ADORA3ADORA2AADORA2BADORA1
SCHEMBL8066488 0.85 MMP13 (0.53) MMP13ADORA3ADORA2AADORA2BADORA1
SCHEMBL8055231 0.84 MMP13 (0.58) MMP13ADORA3ADORA2AADORA2BADORA1
SCHEMBL8071335 0.81 MMP13 (0.58) MMP13CHRM4ALDH1A1LMNAROCK2
SCHEMBL8057403 0.80 MMP13 (0.62) MMP13ADORA3ADORA2AADORA2BADORA1
SCHEMBL3688685 0.79 MMP13 (0.63) MMP13MMP3ROCK2CYP3A4CYP2D6
SCHEMBL3454388 0.78 MMP13 (0.70) MMP13ADORA2AHPGDKDM4EUSP2
SCHEMBL30104666 0.78 ALDH1A1 (0.68) MMP13HPGDKDM4EUSP2ALDH1A1
SCHEMBL8245692 0.78 ALDH1A1 (0.68) MMP13HPGDKDM4EUSP2ALDH1A1
SCHEMBL8069551 0.77 MMP13 (0.61) MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009016498-A1 PYRIMIDINE AND PYRIDINE DERIVATIVES AND THEIR PHARMACEUTICAL USE AND COMPOSITIONS PFIZER INC. (US) 2009-02-05 WO disclosed