SCHEMBL807236

SCHEMBL807236

COc1ccc(CN2CCCCC2)c2ccccc12

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.68
LMNA P02545 4/20 0.68
MAPT P10636 2/20 0.68
HTT P42858 2/20 0.68
ALOX15 P16050 1/20 0.68
SMN1; SMN2 Q16637 1/20 0.68
HSD17B10 Q99714 1/20 0.68
MEN1 O00255 3/20 0.63
KMT2A Q03164 3/20 0.63
ALDH1A1 P00352 2/20 0.63
TSHR P16473 2/20 0.63
TDP1 Q9NUW8 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.50
DRD2 P14416 1/20 0.50
DRD4 P21917 1/20 0.50
HRH2 P25021 1/20 0.50
HRH1 P35367 1/20 0.50
DRD3 P35462 1/20 0.50
SLC2A1 P11166 1/20 0.49
HRH3 Q9Y5N1 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20460271 0.85 KDM4E (0.65) KDM4ELMNAMAPTHTTALOX15
SCHEMBL31618101 0.83 HRH3 (0.68) KDM4ELMNAMAPTHTTALOX15
SCHEMBL24162993 0.82 KDM4E (0.66) KDM4ELMNAMAPTHTTALOX15
SCHEMBL8821609 0.82 LMNA (0.62) KDM4ELMNAMAPTHTTALOX15
SCHEMBL20460351 0.80 ALDH1A1 (0.72) KDM4ELMNAMAPTHTTALOX15
SCHEMBL20460320 0.80 KDM4E (0.67) KDM4ELMNAMAPTHTTALOX15
SCHEMBL3161038 0.80 MEN1 (0.82) KDM4EMEN1KMT2AALDH1A1TSHR
SCHEMBL20460365 0.79 LMNA (0.62) KDM4ELMNAMAPTHTTALOX15
SCHEMBL13284339 0.78 MEN1 (0.79) KDM4EALOX15MEN1KMT2AALDH1A1
SCHEMBL11928962 0.78 CHRM2 (0.72) KDM4ELMNAHTTSMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012036997-A1 FUSED PYRAZOLE DERIVATIVES AS NOVEL ERK INHIBITORS SCHERING CORPORATION (US) 2012-03-22 WO disclosed