SCHEMBL807390

SCHEMBL807390

CCC[C@@H]1CCCN(Cc2cc3ccccc3n2C)C1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.44
MCHR1 Q99705 1/20 0.43
HCRTR1 O43613 1/20 0.40
HCRTR2 O43614 1/20 0.40
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40
OPRL1 P41146 1/20 0.40
HTT P42858 1/20 0.39
MAOA P21397 1/20 0.39
DRD2 P14416 1/20 0.39
DRD1 P21728 1/20 0.39
DRD4 P21917 1/20 0.39
DRD5 P21918 1/20 0.39
DRD3 P35462 1/20 0.39
KDM1A O60341 1/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15084309 0.83 HRH3 (0.48) FAAHMCHR1
SCHEMBL20281637 0.81 TMEM97 (0.48) FAAHMCHR1HCRTR1HCRTR2OPRK1
SCHEMBL15081965 0.80 OPRM1 (0.53) FAAHMCHR1HCRTR1HCRTR2OPRM1
SCHEMBL807593 0.78 FAAH (0.57) FAAHMCHR1HCRTR1HCRTR2OPRM1
SCHEMBL10005899 0.76 FAAH (0.52) FAAHMCHR1
SCHEMBL12513821 0.75 CYP2D6 (0.59) CYP2D6
SCHEMBL10212322 0.75 CYP2D6 (0.59) CYP2D6
SCHEMBL15147442 0.74 FAAH (0.50) FAAHMCHR1
SCHEMBL14375252 0.74 ACHE (0.55) FAAHMCHR1KDM1A
SCHEMBL20281852 0.74 MCHR1 (0.43) FAAHMCHR1OPRK1MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012036997-A1 FUSED PYRAZOLE DERIVATIVES AS NOVEL ERK INHIBITORS SCHERING CORPORATION (US) 2012-03-22 WO disclosed