SCHEMBL807463

SCHEMBL807463

Nc1ccc2c(c1)C1C3=C(C(=O)NC3=O)C2c2cc(N)ccc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.39
CHRNA4 P43681 1/20 0.39
ATM Q13315 1/20 0.37
AKR1B1 P15121 1/20 0.36
CA9 Q16790 3/20 0.34
CA12 O43570 2/20 0.34
DDB1 Q16531 5/20 0.34
CRBN Q96SW2 5/20 0.34
CYP3A4 P08684 3/20 0.33
ALDH1A1 P00352 2/20 0.33
TP53 P04637 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33
PKM P14618 1/20 0.33
HPGD P15428 1/20 0.33
ALOX15 P16050 1/20 0.33
ALOX12 P18054 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10070929 0.75 CYP3A4 (0.47) CHRNB2CHRNA4CA9CA12CYP3A4
SCHEMBL18682060 0.75 CYP3A4 (0.47) CHRNB2CHRNA4CA9CA12CYP3A4
SCHEMBL29636243 0.69 CYP3A4 (0.48) CHRNB2CHRNA4CA9CA12CYP3A4
SCHEMBL807465 0.69 CYP3A4 (0.48) CHRNB2CHRNA4CA9CA12CYP3A4
SCHEMBL29549133 0.69 CYP3A4 (0.48) CHRNB2CHRNA4CA9CA12CYP3A4
SCHEMBL23567922 0.69 CYP3A4 (0.48) CHRNB2CHRNA4CA9CA12CYP3A4
SCHEMBL372282 0.66 ATM (0.58) ATMCA9CA12CYP3A4ALDH1A1
SCHEMBL17789217 0.64 ACHE (0.46) CHRNB2CHRNA4ATMCYP3A4ALDH1A1
Hydrochloric Acid SCHEMBL14890696 0.64 ATM (0.56) ATMCA9CA12CYP3A4ALDH1A1
SCHEMBL22080750 0.63 CA12 (0.41) CHRNB2CHRNA4ATMCA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035327-A1 POLYMERISATION METHOD UNIVERSITY COLLEGE CARDIFF CONSULTANTS LIMITED (GB) 2012-03-22 WO disclosed