SCHEMBL8075290

SCHEMBL8075290

CCCc1ccc(-c2ccc(F)cc2F)cc1.CN[C@H](CS)C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 1/20 0.46
ACE P12821 2/20 0.40
FDFT1 P37268 1/20 0.40
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA12 O43570 1/20 0.39
CA4 P22748 1/20 0.39
CA9 Q16790 1/20 0.39
MMP2 P08253 3/20 0.38
MMP3 P08254 3/20 0.38
MEN1 O00255 3/20 0.38
PTGS1 P23219 3/20 0.38
KMT2A Q03164 3/20 0.38
PTGS2 P35354 2/20 0.38
SLC22A6 Q4U2R8 2/20 0.38
LMNA P02545 2/20 0.38
HPGD P15428 2/20 0.38
HIF1A Q16665 2/20 0.38
AKR1C3 P42330 2/20 0.38
AKR1C2 P52895 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8079610 0.84 MMP2 (0.49) ACEMMP2MMP3MME
SCHEMBL8064698 0.84 MEN1 (0.42) ACECA1CA2MEN1PTGS1
SCHEMBL8079616 0.84 MEN1 (0.42) ACECA1CA2MEN1PTGS1
SCHEMBL9221137 0.79 RARB (0.50) RARBFDFT1CA1CA2MEN1
SCHEMBL8990699 0.78 RARB (0.49) RARBFDFT1CA1CA2MEN1
SCHEMBL8066034 0.77 ACE (0.45) ACEMMP2MEN1KMT2ALMNA
SCHEMBL8080452 0.77 ACE (0.45) ACEMMP2MEN1KMT2ALMNA
SCHEMBL8073254 0.76 ACE (0.45) ACEMMP2MMP3PTGS2KDM4E
SCHEMBL8726493 0.76 RARB (0.48) RARBFDFT1CA1CA2MEN1
SCHEMBL8080420 0.76 SLC6A4 (0.46) ACEMMP2MMP3KMT2APTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6166072-A Amino acid derivatives ALLELIX NEUROSCIENCE, INC. (CA) 2000-12-26 US disclosed
WO-1999034790-A1 GLYCINE TRANSPORT INHIBITORS ALLELIX NEUROSCIENCE, INC. (US) 1999-07-15 WO disclosed