SCHEMBL807646

SCHEMBL807646

Cc1cc(C(=N)C2=C(N)CCN(C(=O)NC3CC(C)CN(Cc4csc5ccccc45)C3)C2)ccn1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.38
PDE2A O00408 1/20 0.34
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
MAPK1 P28482 1/20 0.32
DRD2 P14416 1/20 0.32
DRD4 P21917 1/20 0.32
DRD3 P35462 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL806814 0.79
SCHEMBL15065711 0.69
SCHEMBL15084407 0.69
SCHEMBL807471 0.66
SCHEMBL18360666 0.66 ROCK2 (0.44)
SCHEMBL15084357 0.65 CHRNA7 (0.60) FAAHPDE2AHDAC8HDAC6DRD2
SCHEMBL18360668 0.65 PRMT5 (0.35) FAAHMAPK1
SCHEMBL15065414 0.63
SCHEMBL15065068 0.63 PIP5K1C (0.44)
SCHEMBL14872679 0.62

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012036997-A1 FUSED PYRAZOLE DERIVATIVES AS NOVEL ERK INHIBITORS SCHERING CORPORATION (US) 2012-03-22 WO disclosed