SCHEMBL807721

SCHEMBL807721

COc1ccc2nc(Nc3cc(CN4CCOCC4)cc(N[C@H]4CCN(C(=O)OC(C)(C)C)C4)n3)sc2c1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.49
SCD O00767 1/20 0.44
DYRK1A Q13627 1/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
LRRK2 Q5S007 1/20 0.43
WNT3A P56704 1/20 0.43
CASR P41180 1/20 0.43
USP2 O75604 1/20 0.42
MAPT P10636 1/20 0.42
CLK1 P49759 1/20 0.42
MAPK10 P53779 1/20 0.42
LCK P06239 2/20 0.42
AURKB Q96GD4 3/20 0.42
ITK Q08881 2/20 0.41
TBK1 Q9UHD2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL807714 0.90 ITK (0.46) NPC1RAB9ALCKITKTBK1
SCHEMBL10285559 0.89 KMT2A (0.51) KMT2ASCDNPC1RAB9ALRRK2
SCHEMBL807926 0.84 ITK (0.59) LCKAURKBITKTBK1
SCHEMBL807541 0.80 ITK (0.55) LCKAURKBITKTBK1
SCHEMBL23608014 0.78 BTK (0.42) ITKTBK1
SCHEMBL21792649 0.78 BTK (0.42) ITKTBK1
SCHEMBL2677855 0.77 NPC1 (0.54) KMT2ASCDDYRK1ANPC1RAB9A
SCHEMBL2677854 0.77 NPC1 (0.54) KMT2ASCDDYRK1ANPC1RAB9A
SCHEMBL29261762 0.76 BTK (0.41) ITKTBK1
SCHEMBL21792590 0.76 BTK (0.41) ITKTBK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035055-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-22 WO disclosed